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13 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of 5-benzyl-3-phenyl-4,5-dihydroisoxazoles and 5-benzyl-3-phenyl-1,4,2-dioxazoles as potent firefly luciferase inhibitors.EBI
University of Eastern Finland
Synthesis of an N-acyl sulfamate analog of luciferyl-AMP: a stable and potent inhibitor of firefly luciferase.EBI
Connecticut College
Identification of a naturally occurring quinazolin-4(3H)-one firefly luciferase inhibitor.EBI
Merlion Pharmaceuticals
Discovery, synthesis, and biological evaluation of novel SMN protein modulators.EBI
National Human Genome Research Institute
A basis for reduced chemical library inhibition of firefly luciferase obtained from directed evolution.EBI
National Institutes of Health
False positives in a reporter gene assay: identification and synthesis of substituted N-pyridin-2-ylbenzamides as competitive inhibitors of firefly luciferase.EBI
Leiden/Amsterdam Center For Drug Research
Kinetic Target-Guided Synthesis: Reaching the Age of Maturity.EBI
Univ. Lille
Discovery of an isocoumarin analogue that modulates neuronal functions via neurotrophin receptor TrkB.EBI
Indian Institute of Technology Madras
Identification and synthesis of substituted pyrrolo[2,3-d]pyrimidines as novel firefly luciferase inhibitors.EBI
Chinese Academy of Sciences
Characterization of chemical libraries for luciferase inhibitory activity.EBI
National Human Genome Research Institute
Identification of fused pyrimidines as interleukin 17 secretion inhibitors.EBI
Norwegian University of Science and Technology
Tryptophan hydroxylase inhibitor and pharmaceutical composition including sameBDB
Gwangju Institute of Science and Technology
A TMPRSS2 inhibitor acts as a pan-SARS-CoV-2 prophylactic and therapeutic.BDB
University of British Columbia