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BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 698K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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38 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Spirocyclic 2,3-dihydro-7-azaindole compounds and uses thereofBDB
Genentech
CRYSTALLINE FORMS OF (4S)-24-CHLORO-4-ETHYL-73-FLUORO-35-METHOXY-32,5-DIOXO-14-(TRIFLUORO-METHYL)-32H-6-AZA-3(4,1)-PYRIDINA-1(1)-[1,2,3]TRIAZOLA-2(1,2),7(1)-DIBENZENAHEPTAPHANE-74-CARBOXAMIDEBDB
Bayer Aktiengesellschaft
Nitrogen-Containing Heterocyclic Compound, Pharmaceutical Compositions thereof and Use thereofBDB
280 Bio
Imino sulfanone inhibitors of ENPP1BDB
Volastra Therapeutics
Therapeutic agent for non-motor symptoms associated with Parkinson's diseaseBDB
Sumitomo Pharma
Imidazole and triazole containing bicyclic compounds as JAK inhibitorsBDB
Theravance Biopharma R&D Ip
Tetrahydro-imidazo quinoline compositions as CBP/P300 inhibitorsBDB
Forma Therapeutics
Macrocyclic compounds that inhibit MCL-1 proteinBDB
Amgen
Fused imidazo-piperidine JAK inhibitorsBDB
Theravance Biopharma R&D Ip
Macrocyclic compounds for treatment of medical disordersBDB
Achillion Pharmaceuticals
CXCR7 antagonistsBDB
Chemocentryx
Toll-like receptor 7 (TLR7) agonists having a tricyclic moiety, conjugates thereof, and methods and uses thereforBDB
Bristol-Myers Squibb Companay
Oxadiazolones as transient receptor potential channel inhibitorsBDB
Genentech
Epoxyketone compounds for enzyme inhibitionBDB
Centrax International
Condensed-ring pyrimidylamino derivative, preparation method therefor, and intermediate, pharmaceutical composition and applications thereofBDB
Guangzhou Maxinovel Pharmaceuticals
[4-(1,3,3-trimethyl-2-oxo-3,4-dihydro-1H-quinoxalin-7-yl)phenoxy]ethyloxy compound or salt thereofBDB
Santen Pharmaceutical
Pyrrolo[2,3-d]pyrimidine compound or salt thereofBDB
Taiho Pharmaceutical
Heteroaryl substituted pyrrolotriazine amine compounds as PI3K inhibitorsBDB
Bristol-Myers Squibb
Protein kinase C inhibitors and methods of their useBDB
Novartis
Alpha-carbolines for the treatment of cancerBDB
Universita Degli Studi Di Milano—Bicocca
Indole and indazole compounds that activate AMPKBDB
Pfizer
Carbonic anhydrase inhibitors: in vitro inhibition of a isoforms (hCA I, hCA II, bCA III, hCA IV) by flavonoids.BDB
Ondokuz Mayis University
Bicyclic substituted pyrimidine compoundsBDB
Xuanzhu Pharma
Compositions and methods for the treatment of malariaBDB
Saint Louis University
5-HT3 receptor antagonistsBDB
Takeda Pharmaceutical
Optically pure benzyl-4-chlorophenyl-C-glucoside derivativeBDB
Xuanzhu Pharma
Triazolopyridinone PDE10 inhibitorsBDB
Merck Sharp & Dohme
Functional reversal of (-)-Stepholidine analogues by replacement of benzazepine substructure using the ring-expansion strategy.BDB
Fudan University
Tricyclic heterocyclic compoundsBDB
Bristol-Myers Squibb
Compounds and methods for purification of serine proteasesBDB
Portola Pharmaceuticals
Inhibition of memapsin 1 cleavage in the treatment of diabetesBDB
Oklahoma Medical Research Foundation
Selective caspase inhibitors and uses thereofBDB
Novagenesis Foundation
Discovery of isoalloxazine derivatives as a new class of potential anti-Alzheimer agents and their synthesis.BDB
The M. S. University of Baroda
Pyridinedione carboxamide inhibitors of endothelial lipaseBDB
Bristol-Myers Squibb
Aminopyrazole derivativeBDB
Chugai Seiyaku Kabushiki Kaisha
Thieno[3,2-C]pyridine kinase inhibitors with improved CYP safety profileBDB
Abbvie
Photoaffinity labeling of the Ah receptor.BDB
University of Wisconsin
Somatostatin and its receptor family.BDB
Royal Victoria Hospital