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9 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Structure guided design of a series of sphingosine kinase (SphK) inhibitors.EBI
Amgen
Design, synthesis and biological activity of sphingosine kinase 2 selective inhibitors.EBI
Virginia Tech
Development of amidine-based sphingosine kinase 1 nanomolar inhibitors and reduction of sphingosine 1-phosphate in human leukemia cells.EBI
University of Virginia
Rational design of SphK inhibitors using crystal structures aided by computer.EBI
Shandong First Medical University & Shandong Academy of Medical Sciences
Discovery of In Vivo Active Sphingosine-1-phosphate Transporter (Spns2) Inhibitors.EBI
Virginia Tech
Discovery of a Small Side Cavity in Sphingosine Kinase 2 that Enhances Inhibitor Potency and Selectivity.EBI
Virginia Tech
Transforming Sphingosine Kinase 1 Inhibitors into Dual and Sphingosine Kinase 2 Selective Inhibitors: Design, Synthesis, and in Vivo Activity.EBI
University of Virginia
Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B.EBI
Kyoto University
Imidamide sphingosine kinase inhibitorsBDB
University of Virginia Patent Foundation