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17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis and evaluation of novel (18)F-labeled spirocyclic piperidine derivatives ass1 receptor ligands for positron emission tomography imaging.EBI
Key Laboratory of Radiopharmaceuticals Beijing Normal University
Stereoselective synthesis of a new class of potent and selective inhibitors of human¿8,7-sterol isomerase.EBI
Ludwig-Maximilians University
New positron emission tomography (PET) radioligand for imagings-1 receptors in living subjects.EBI
Stanford University
Exploring the importance of piperazine N-atoms for sigma(2) receptor affinity and activity in a series of analogs of 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28).EBI
Universita Degli Studi Di Bari
Novel 4-(4-aryl)cyclohexyl-1-(2-pyridyl)piperazines as Delta(8)-Delta(7) sterol isomerase (emopamil binding protein) selective ligands with antiproliferative activity.EBI
Universita Degli Studi Di Bari
Design and evaluation of naphthol- and carbazole-containing fluorescent sigma ligands as potential probes for receptor binding studies.EBI
University of Bari Aldo Moro
Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma(1) receptor.EBI
University of Bari Aldo Moro
Discovery of high-affinity ligands of sigma1 receptor, ERG2, and emopamil binding protein by pharmacophore modeling and virtual screening.EBI
University of Innsbruck
Synthesis of chiral 1-[omega-(4-chlorophenoxy)alkyl]-4-methylpiperidines and their biological evaluation at sigma1, sigma2, and sterol delta8-delta7 isomerase sites.EBI
University of Bari Aldo Moro
Synthesis, radiofluorination and pharmacological evaluation of a fluoromethyl spirocyclic PET tracer for centrals1 receptors and comparison with fluoroalkyl homologs.EBI
Institute of Radiopharmacy
Synthesis and binding assays of novel 3,3-dimethylpiperidine derivatives with various lipophilicities ass¿? receptor ligands.EBI
University of Bari Aldo Moro
Synthesis and biological evaluation of novel 4-benzylpiperazine ligands for sigma-1 receptor imaging.EBI
Key Laboratory of Radiopharmaceuticals (Beijing Normal University)
Emopamil-Binding Protein Inhibitors for Treating Multiple Sclerosis.EBI
Smith, Gambrell & Russell
Emopamil-Binding Protein Inhibitors for Treating Multiple Sclerosis.EBI
Smith, Gambrell & Russell
Emopamil-Binding Protein Inhibitors for Treating Multiple Sclerosis.EBI
Smith, Gambrell & Russell
A perspective on medicinal chemistry approaches towards adenomatous polyposis coli and Wnt signal based colorectal cancer inhibitors.EBI
Gitam (Deemed To Be University)
PRMT5 INHIBITOR AND THE USE THEREOFBDB
Cytosinlab Therapeutics