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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 748K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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26 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Iridinesulfonamide compound and use method thereofBDB
Chia Tai Tianqing Pharmaceutical Group
Substituted 6,11-dihydro-5H-benzo[B]carbazoles as inhibitors of ALK and SRPKBDB
Dana-Farber Cancer Institute
Immunomodulator compounds and methods of useBDB
Incyte
Selective estrogen receptor degradersBDB
Eli Lilly
Substituted bicyclic dihydropyrimidinones and their use as inhibitors of neutrophil elastase activityBDB
Boehringer Ingelheim International
Selective CYP11B1 inhibitors for the treatment of cortisol dependent diseasesBDB
Universitaet Des Saarlandes Campus Saarbruecken
Urease inhibitors from Indigofera gerardiana Wall.BDB
Khyber Medical College
Nitrogen-containing bicyclic aromatic heterocyclic compoundBDB
Astellas Pharma
Imidazopyridin-2-one derivativesBDB
Merck Sharp & Dohme
Phenylpyridine derivative and drug containing sameBDB
Kowa
In vivo anti-inflammatory activity and docking study of newly synthesized benzimidazole derivatives bearing oxadiazole and morpholine rings.BDB
Jamia Hamdard (Hamdard University)
Acyl piperidine inhibitors of soluble epoxide hydrolaseBDB
University of California
Histone deacetylase 7 promotes Toll-like receptor 4-dependent proinflammatory gene expression in macrophages.BDB
University of Queensland
Oligomer-opioid agonist conjugatesBDB
Nektar Therapeutics
Tropomyosin-related kinase (TRK) inhibitorsBDB
Genzyme
Proline sulfonamide derivatives as orexin receptor antagonistsBDB
Actelion Pharmaceuticals
Multifunctional radical quenchers and their usesBDB
Arizona Board of Regents, A Body Corporate of The State of Arizona Acting For and On Behalf of Arizona State University
Buprenorphine analogsBDB
Purdue Pharma
Benzodioxole piperidine compoundsBDB
Hoffmann-La Roche
Structure-based design and solid-phase parallel synthesis of phosphorylated nonpeptides to explore hydrophobic binding at the Src SH2 domain.BDB
Ariad Pharmaceuticals
Steady-state kinetic mechanism of Ras farnesyl:protein transferase.BDB
Merck Research Laboratories
Reaction of the molybdenum- and copper-containing carbon monoxide dehydrogenase from Oligotropha carboxydovorans with quinones.BDB
University of California Riverside
N-(3-lodoprop-2E-enyl)-2beta-carbomethoxy-3beta-(3',4'-dichloro phenyl)nortropane (beta-CDIT), a tropane derivative: pharmacological characterization as a specific ligand for the dopamine transporter in the rodent brain.BDB
University of Tours
Displacement of DL-[3H]-2-amino-4-phosphonobutanoic acid ( [3H]APB) binding with methyl-substituted APB analogues and glutamate agonists.BDB
University of Minnesota
Characterization of flufylline, fluprofylline, ritanserin, butanserin and R 56413 with respect to in-vivo alpha 1-,alpha 2- and 5-HT2-receptor antagonism and in-vitro affinity for alpha 1-,alpha 2- and 5-HT2-receptors: comparison with ketanserin.BDB
TBA
 
Human Plasma Lecithin-Cholesterol AcyltransferaseBDB
Dalhousie University