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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 748K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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17 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of the Irreversible Covalent FGFR Inhibitor 8-(3-(4-Acryloylpiperazin-1-yl)propyl)-6-(2,6-dichloro-3,5-dimethoxyphenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8H)-one (PRN1371) for the Treatment of Solid Tumors.EBI
Principia Biopharma
Compositions and methods for treating CNS disordersBDB
Sage Therapeutics
Pyrazole[1,5-a] pyrimidine derivatives as kinase JAK inhibitorsBDB
Celon Pharma
Substituted N′-hydroxycarbamimidoyl-1,2,5-oxadiazole compounds as indoleamine 2,3-dioxygenase IDO inhibitorsBDB
Merck Sharp & Dohme
Substituted indole Mcl-1 inhibitorsBDB
Vanderbilt University
Tetrahydroimidazo(1,5-D)[1,4]oxazepine derivativeBDB
Eisai R&D Management
Acid ceramidase inhibitors and their use as medicamentsBDB
Fondazione Istituto Italiano Di Technologia
Inhibition of the ß-class carbonic anhydrases from Mycobacterium tuberculosis with carboxylic acids.BDB
Universit�� Degli Studi Di Firenze
 
Synthesis, biological evaluation and molecular modeling study of new (1,2,4-triazole or 1,3,4-thiadiazole)-methylthio-derivatives of quinazolin-4(3H)-one as DHFR inhibitorsBDB
Future University
Process for preparing spirocyclic cyclohexane compounds, compositions containing such compounds and method of using such compoundsBDB
Gruenenthal
Indolizine compounds, a process for their preparation and pharmaceutical compositions containing themBDB
Les Laboratoires Servier
Triazole double-headed ribonucleosides as inhibitors of eosinophil derived neurotoxin.BDB
University of Thessaly
Acetylcholinesterase/butyrylcholinesterase inhibition activity of some new carbacylamidophosphate derivatives.BDB
Tarbiat Modares University
Design and synthesis of morpholine derivatives. SAR for dual serotonin & noradrenaline reuptake inhibition.BDB
Pfizer
The binding of L-[3H]nicotine to a single class of high affinity sites in rat brain membranes.BDB
R. J. Reynolds Tobacco
Allosteric non-bisphosphonate FPPS inhibitors identified by fragment-based discovery.BDB
Novartis Institutes For Biomedical Research