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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.5M data for 737K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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10 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Small molecule direct inhibitors of KEAP1-NRF2 protein-protein interactionBDB
The State University of New Jersey
HETEROARYL AMIDES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOFBDB
Merck Sharp & Dohme
Antitumor Activity of Cytotoxic Cyclooxygenase-2 Inhibitors.BDB
Vanderbilt Institute of Chemical Biology, Vanderbilt University School of Medicine
Epiblastin A Induces Reprogramming of Epiblast Stem Cells Into Embryonic Stem Cells by Inhibition of Casein Kinase 1.BDB
Max Planck Institute of Molecular Physiology
Quinoxaline carboxamide derivatives as protein tyrosine kinase inhibitorsBDB
Novartis
Evidence for the preferential involvement of 5-HT2A serotonin receptors in stress- and drug-induced dopamine release in the rat medial prefrontal cortex.BDB
Case Western Reserve University
Elucidation of vasoactive intestinal peptide pharmacophore for VPAC(1) receptors in human, rat, and guinea pig.BDB
National Institutes of Health
OPC-28326, a selective femoral vasodilator, is an alpha2C-adrenoceptor-selective antagonist.BDB
Otsuka Maryland Research Institute
A quick diversity-oriented amide-forming reaction to optimize P-subsite residues of HIV protease inhibitors.BDB
The Scripps Research Institute