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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.5M data for 737K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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25 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Indole and azaindole inhibitors of pad enzymesBDB
Bristol-Myers Squibb
Aryl-phosphorus-oxygen compound as EGFR kinase inhibitorBDB
Chia Tai Tianqing Pharmaceutical Group
Triple combination of pure 5-HT6 receptor antagonists, acetylcholinesterase inhibitors and NMDA receptor antagonistBDB
Suven Life Sciences
Compositions and methods for treating parasitic diseasesBDB
University of California
LRRK2 inhibitors and methods of making and using the sameBDB
Dana-Farber Cancer Institute
Amido spirocyclic amide and sulfonamide derivativesBDB
Forma Tm
1-cyano-pyrrolidine compounds as USP30 inhibitorsBDB
Mission Therapeutics
Covalent small molecule DCN1 inhibitors and therapeutic methods using the sameBDB
University of Michigan
Substituted indoles as modulators of ROR-gammaBDB
Vitae Pharmaceuticals
N-Methylbenzimidazoles as mIDH1 inhibitorsBDB
Bayer Pharma Aktiengesellschaft
Thienopyrimidine compoundsBDB
Hoffmann-La Roche
Arylpyrrolopyridine derived compounds as LRRK2 inhibitorsBDB
H. Lundbeck
Synthesis and dual D2 and 5-HT1A receptor binding affinities of 5-piperidinyl and 5-piperazinyl-1H-benzo[d]imidazol-2(3H)-ones.BDB
King Fahd University of Petroleum & Minerals
Substituted imidazo[1,2-b]pyridazines as protein kinase inhibitorsBDB
Tolero Pharmaceuticals
New hybrid molecules combining benzothiophene or benzofuran with rhodanine as dual COX-1/2 and 5-LOX inhibitors: Synthesis, biological evaluation and docking study.BDB
Alexandria University
Heteroaryl linked quinolinyl modulators of RORγtBDB
Janssen Pharmaceutica
Amino-substituted imidazopyridazinesBDB
Bayer Pharma Aktiengesellschaft
Bicarbocyclic and tricarbocyclic ethynyl derivatives and uses of sameBDB
H. Lundbeck
Novel biphenyl bis-sulfonamides as acetyl and butyrylcholinesterase inhibitors: Synthesis, biological evaluation and molecular modeling studies.BDB
Government College University
Cycloalkane carboxylic acid derivatives as CXCR3 receptor antagonistsBDB
Sanofi
2-heteroaryl carboxamidesBDB
Bayer Intellectual Property
Cyclohexane-1,2′-naphthalene-1′,2″-imidazol compounds and their use as BACE inhibitorsBDB
Astrazeneca
Inhibition of fucosyltransferase VII by gallic acid and its derivatives.BDB
Schering-Plough Research Institute
Pharmacological characterization of KUR-1246, a selective uterine relaxant.BDB
Kissei Pharmaceutical
2-cyano-3-cyclopropyl-3-hydroxy-N-aryl-thioacrylamide derivativesBDB
Algiax Pharmaceuticals