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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 748K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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9 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of CRN04894: A Novel Potent Selective MC2R Antagonist.EBI
Crinetics Pharmaceuticals
Discovery of Paltusotine (CRN00808), a Potent, Selective, and Orally Bioavailable Non-peptide SST2 Agonist.EBI
Crinetics Pharmaceuticals
Discovery of 4-(3-aminopyrrolidinyl)-3-aryl-5-(benzimidazol-2-yl)-pyridines as potent and selective SST5 agonists for the treatment of congenital hyperinsulinism.EBI
Crinetics Pharmaceuticals
Discovery of substituted 3H-pyrido[2,3-d]pyrimidin-4-ones as potent, biased, and orally bioavailable sst2 agonist.EBI
Crinetics Pharmaceuticals
Heterocyclic compounds as kinase inhibitorsBDB
Nuvation Bio
OXA-Diazaspiro compounds having activity against painBDB
Esteve Pharmaceuticals
1,3-dihydroxy-phenyl derivatives useful as immunomodulatorsBDB
Bristol-Meyers Squibb
Protein kinase inhibitors (variants), use thereof in treating oncological diseases and a pharmaceutical composition based thereonBDB
Obshchestvo S Ogranichennoy Otvetstvennostyou “Fusion Pharma”
PET Imaging agentsBDB
Novartis