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BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 698K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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14 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis, characterization, and optimization for in vivo delivery of a nonselective isopeptidase inhibitor as new antineoplastic agent.EBI
University of Trieste
X-ray structural and biological evaluation of a series of potent and highly selective inhibitors of human coronavirus papain-like proteases.EBI
Purdue University
Spongiacidin C, a pyrrole alkaloid from the marine sponge Stylissa massa, functions as a USP7 inhibitor.EBI
Kumamoto University
Discovery and Characterization of BAY-805, a Potent and Selective Inhibitor of Ubiquitin-Specific Protease USP21.EBI
Bayer
Recent advances in the development of ubiquitin-specific-processing protease 7 (USP7) inhibitors.EBI
Zhengzhou University
Structure-Activity Relationship of USP5 Inhibitors.EBI
University of Toronto
Discovery of Potent Small-Molecule USP8 Inhibitors for the Treatment of Breast Cancer through Regulating ERα Expression.EBI
China Pharmaceutical University
Discovery of Potent OTUB1/USP8 Dual Inhibitors Targeting Proteostasis in Non-Small-Cell Lung Cancer.EBI
Fudan University
Discovery of Potent, Selective, and Orally Bioavailable Inhibitors of USP7 with In Vivo Antitumor Activity.EBI
Rapt Therapeutics
Advances in Discovering Deubiquitinating Enzyme (DUB) Inhibitors.EBI
Dana-Farber Cancer Institute
Identification of small-molecule inhibitors of USP2a.EBI
Jagiellonian University
Chemical Approaches to Intervening in Ubiquitin Specific Protease 7 (USP7) Function for Oncology and Immune Oncology Therapies.EBI
Progenra
Development of a highly reliable assay for ubiquitin-specific protease 2 inhibitors.EBI
Shanghai Jiao Tong University
Guanidine compoundBDB
Astellas Pharma