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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Compounds and compositions as RAF kinase inhibitorsBDB
Novartis
Opioid agonists and uses thereofBDB
Nektar Therapeutics
Thiazoles as modulators of RORγtBDB
Janssen Pharmaceutica
Keto-imidazopyridine derivatives as RORc modulatorsBDB
Genentech
2-(morpholin-4-yl)-1,7-naphthyridinesBDB
Bayer Pharma Aktiengesellschaft
Selective glycosidase inhibitors and uses thereofBDB
Alectos Therapeutics
BTK InhibitorsBDB
Merck Sharp & Dohme
Macrocyclic compounds as Trk kinase inhibitorsBDB
Array Biopharma
Substituted aza-bicyclic imidazole derivatives useful TRPM8 receptor modulatorsBDB
Janssen Pharmaceutica
Non-nucleoside reverse transcriptase inhibitorsBDB
Merck Sharp & Dohme
Discovery of potent antagonists of the antiapoptotic protein XIAP for the treatment of cancer.BDB
Abbott Laboratories
Structure-based design of caspase-1 inhibitor containing a diphenyl ether sulfonamide.BDB
Pfizer
New anilinophthalazines as potent and orally well absorbed inhibitors of the VEGF receptor tyrosine kinases useful as antagonists of tumor-driven angiogenesis.BDB
Novartis Pharmaceuticals
Tyrosine kinase inhibitors. 18. 6-Substituted 4-anilinoquinazolines and 4-anilinopyrido[3,4-d]pyrimidines as soluble, irreversible inhibitors of the epidermal growth factor receptor.BDB
University of Auckland
2-Pyridinone derivatives: a new class of nonnucleoside, HIV-1-specific reverse transcriptase inhibitors.BDB
Merck Sharp and Dohme Research Laboratories
Nonpeptidic HIV protease inhibitors possessing excellent antiviral activities and therapeutic indices. PD 178390: a lead HIV protease inhibitor.BDB
Parke-Davis Pharmaceutical Research
Phenethylthiazolylthiourea (PETT) compounds as a new class of HIV-1 reverse transcriptase inhibitors. 2. Synthesis and further structure-activity relationship studies of PETT analogs.BDB
Eli Lilly
Design and synthesis of HIV protease inhibitors. Variations of the carboxy terminus of the HIV protease inhibitor L-682,679.BDB
Merck Sharp and Dohme Research Laboratories