37 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Coumarin sulfonates: New alkaline phosphatase inhibitors; in vitro and in silico studies.
University of Karachi
Synthesis, alkaline phosphatase inhibition studies and molecular docking of novel derivatives of 4-quinolones.
Universit£T Rostock
2-Alkoxy-3-(sulfonylarylaminomethylene)-chroman-4-ones as potent and selective inhibitors of ectonucleotidases.
Forman Christian College (A Chartered University)
Diarylsulfonamides and their bioisosteres as dual inhibitors of alkaline phosphatase and carbonic anhydrase: Structure activity relationship and molecular modelling studies.
Forman Christian College (A Chartered University)
Design, synthesis and evaluation of benzoisothiazolones as selective inhibitors of PHOSPHO1.
Sanford-Burnham Medical Research Institute
Identification of a selective inhibitor of murine intestinal alkaline phosphatase (ML260) by concurrent ultra-high throughput screening against human and mouse isozymes.
Sanford-Burnham Medical Research Institute
Identification of novel chromone based sulfonamides as highly potent and selective inhibitors of alkaline phosphatases.
Forman Christian College (A Chartered University)
Alkaline phosphatase inhibition by a series of pyrido[2,1-b]quinazolines: A possible relationship with cromolyn-like antiallergy activity.
TBA
Synthesis and evaluation of thiophenyl derivatives as inhibitors of alkaline phosphatase.
University of Lyon 1
Design and synthesis of selective inhibitors of placental alkaline phosphatase.
Human Biomolecular Research Institute
Synthesis and evaluation of benzo[b]thiophene derivatives as inhibitors of alkaline phosphatases.
University of Lyon
Discovery and validation of a series of aryl sulfonamides as selective inhibitors of tissue-nonspecific alkaline phosphatase (TNAP).
Institute For Medical Research
Design and synthesis of pyrazole derivatives as potent and selective inhibitors of tissue-nonspecific alkaline phosphatase (TNAP).
Institute For Medical Research
Targeting ecto-5'-nucleotidase: A comprehensive review into small molecule inhibitors and expression modulators.
Federal University of Rio Grande Do Sul
Specific Inhibitor of Placental Alkaline Phosphatase Isolated from a DNA-Encoded Chemical Library Targets Tumor of the Female Reproductive Tract.
Swiss Federal Institute of Technology (Eth Z£Rich)
A comparison of phosphonothioic acids with phosphonic acids as phosphatase inhibitors.
Utah State University
Exploration of carboxy pyrazole derivatives: Synthesis, alkaline phosphatase, nucleotide pyrophosphatase/phosphodiesterase and nucleoside triphosphate diphosphohydrolase inhibition studies with potential anticancer profile.
Quaid-I-Azam University
Hybrid compounds from chalcone and 1,2-benzothiazine pharmacophores as selective inhibitors of alkaline phosphatase isozymes.
University of Auckland
2-Substituted 7-trifluoromethyl-thiadiazolopyrimidones as alkaline phosphatase inhibitors. Synthesis, structure activity relationship and molecular docking study.
Universit£T Rostock
Discovery of 5-((5-chloro-2-methoxyphenyl)sulfonamido)nicotinamide (SBI-425), a potent and orally bioavailable tissue-nonspecific alkaline phosphatase (TNAP) inhibitor.
Sanford Burnham Prebys Medical Discovery Institute
Compounds useful as inhibitors of indoleamine 2,3-dioxygenase and/or tryptophan dioxygenase
University Of Texas
Substituted oxopyridine derivatives and use thereof in the treatment of cardiovascular disorders
Bayer Pharma Aktiengesellschaft
Tetrahydronaphthyridine, benzoxazine, aza-benzoxazine and related bicyclic compounds for inhibition of RORgamma activity and the treatment of disease
Lycera
Meta-substituted phenyl sulfonyl amides of secondary amino acid amides, the production thereof, and use thereof as matriptase inhibitors
The Medicines Company (Leipzig)
Identification and Characterization of a New Chemotype of Noncovalent SENP Inhibitors.
Beckman Research Institute of The City of Hope
A refined pharmacophore identifies potent 4-amino-7-chloroquinoline-based inhibitors of the botulinum neurotoxin serotype A metalloprotease.
National Cancer Institute At Frederick
Identification of a potent botulinum neurotoxin a protease inhibitor using in situ lead identification chemistry.
The Scripps Research Institute
An in vitro and in vivo disconnect uncovered through high-throughput identification of botulinum neurotoxin A antagonists.
The Scripps Research Institute
N-Acylthiadiazolines, a new class of liver X receptor agonists with selectivity for LXRbeta.
Gnf
Discovery of the HCV NS3/4A protease inhibitor (1R,5S)-N-[3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3- [2(S)-[[[(1,1-dimethylethyl)amino]carbonyl]amino]-3,3-dimethyl-1-oxobutyl]- 6,6-dimethyl-3-azabicyclo[3.1.0]hexan-2(S)-carboxamide (Sch 503034) II. Key steps in structure-based optimization.
Schering-Plough Research Institute