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BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 698K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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8 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of 7-aminofuro[2,3-c]pyridine inhibitors of TAK1: optimization of kinase selectivity and pharmacokinetics.EBI
Osi Pharmaceuticals
Discovery and optimization of 7-aminofuro[2,3-c]pyridine inhibitors of TAK1.EBI
Osi Pharmaceuticals
Oxindole derivatives as inhibitors of TAK1 kinase.EBI
Myrexis
Discovery of 2,4-1EBI
Zobio
Synthesis and anti-tumor activity of imidazopyrazines as TAK1 inhibitors.EBI
Chung-Ang University
Discovery of 7H-pyrrolo[2,3-d]pyrimidine derivatives as selective covalent irreversible inhibitors of interleukin-2-inducible T-cell kinase (Itk).EBI
Peking University
Heterobicyclic N-aminophenyl-amides as inhibitors of histone deacetylaseBDB
Rodin Therapeutics
Benzonitrile derivatives as kinase inhibitorsBDB
Merck Patent