22 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Ynamide Click chemistry in development of triazole VEGFR2 TK modulators.
University of Strasburg
Discovery of Potent Inhibitors of Schistosoma mansoni NAD¿ Catabolizing Enzyme.
University of Strasburg
Selective nonpeptidic fluorescent ligands for oxytocin receptor: design, synthesis, and application to time-resolved FRET binding assay.
University of Strasburg
Catechol-rhodanine derivatives: Specific and promiscuous inhibitors of Escherichia coli deoxyxylulose phosphate reductoisomerase (DXR).
University of Strasburg
Structure-activity relationship studies toward the discovery of selective apelin receptor agonists.
University of Strasburg
Design, synthesis and biological evaluation of novel tetrahydroacridine pyridine- aldoxime and -amidoxime hybrids as efficient uncharged reactivators of nerve agent-inhibited human acetylcholinesterase.
University of Strasburg
Synthesis and biological properties of thiazole-analogues of pyochelin, a siderophore of Pseudomonas aeruginosa.
University of Strasburg
Design, synthesis, and molecular modelling of pyridazinone and phthalazinone derivatives as protein kinases inhibitors.
University of Strasburg
Fluorescent derivatives of AC-42 to probe bitopic orthosteric/allosteric binding mechanisms on muscarinic M1 receptors.
University of Strasburg
Selective fluorescent nonpeptidic antagonists for vasopressin V2 GPCR: application to ligand screening and oligomerization assays.
University of Strasburg
Methylation of imidazoline related compounds leads to loss ofa2-adrenoceptor affinity. Synthesis and biological evaluation of selective I1 imidazoline receptor ligands.
University of Strasburg
Growth inhibition of Mycobacterium smegmatis by prodrugs of deoxyxylulose phosphate reducto-isomerase inhibitors, promising anti-mycobacterial agents.
University of Strasburg
Subtlety of the structure-affinity and structure-efficacy relationships around a nonpeptide oxytocin receptor agonist.
University of Strasburg
Reactive derivatives for affinity labeling in the ifenprodil site of NMDA receptors.
University of Strasburg
New PDE4 inhibitors based on pharmacophoric similarity between papaverine and tofisopam.
University of Strasburg
Synthesis and biological evaluation of desmethylveramiline, a micromolar Hedgehog inhibitor.
University of Strasburg
Cysteine mapping in conformationally distinct kinase nucleotide binding sites: application to the design of selective covalent inhibitors.
University of Strasburg
Heterocyclic bis-cations as starting hits for design of inhibitors of the bifunctional enzyme histidine-containing protein kinase/phosphatase from Bacillus subtilis.
University of Strasburg
