44 articles for thisTarget
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Xanthine oxidase inhibitory activity of nicotino/isonicotinohydrazides: A systematic approach from in vitro, in silico to in vivo studies.
University of Karachi
Coumarin sulfonates: New alkaline phosphatase inhibitors; in vitro and in silico studies.
University of Karachi
Biology-oriented drug synthesis (BIODS): In vitroß-glucuronidase inhibitory and in silico studies on 2-(2-methyl-5-nitro-1H-imidazol-1-yl)ethyl aryl carboxylate derivatives.
University of Karachi
Thiadiazole derivatives as New Class ofß-glucuronidase inhibitors.
University of Karachi
Synthesis of diethyl 4-substituted-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylates as a new series of inhibitors against yeasta-glucosidase.
University of Karachi
Synthesis andß-glucuronidase inhibitory activity of 2-arylquinazolin-4(3H)-ones.
University of Karachi
Evaluation of bisindole as potentß-glucuronidase inhibitors: synthesis and in silico based studies.
University of Karachi
Fungal transformation of cedryl acetate anda-glucosidase inhibition assay, quantum mechanical calculations and molecular docking studies of its metabolites.
University of Karachi
3D-QSAR CoMFA studies on bis-coumarine analogues as urease inhibitors: a strategic design in anti-urease agents.
University of Karachi
Identification of acridinyl hydrazides as potent aspartic protease inhibitors.
University of Karachi
New benzimidazole derivatives as antiplasmodial agents and plasmepsin inhibitors: synthesis and analysis of structure-activity relationships.
University of Karachi
Methylenebissantin: a rare methylene-bridged bisflavonoid from Dodonaea viscosa which inhibits Plasmodium falciparum enoyl-ACP reductase.
University of Karachi
1,3,4-Oxadiazole-2(3H)-thione and its analogues: a new class of non-competitive nucleotide pyrophosphatases/phosphodiesterases 1 inhibitors.
University of Karachi
Microbial transformation and butyrylcholinesterase inhibitory activity of (-)-caryophyllene oxide and its derivatives.
University of Karachi
New triterpenoid alkaloid cholinesterase inhibitors from Buxus hyrcana.
University of Karachi
Isolation and cholinesterase-inhibition studies of sterols from Haloxylon recurvum.
University of Karachi
Synthesis and urease inhibitory potential of benzophenone sulfonamide hybrid in vitro and in silico.
University of Karachi
Synthesis of benzotriazoles derivatives and their dual potential as α-amylase and α-glucosidase inhibitors in vitro: Structure-activity relationship, molecular docking, and kinetic studies.
University of Karachi
Microwave-Assisted Organic Synthesis, structure-activity relationship, kinetics and molecular docking studies of non-cytotoxic benzamide derivatives as selective butyrylcholinesterase inhibitors.
University of Karachi
Synthesis of novel inhibitors of β-glucuronidase based on benzothiazole skeleton and study of their binding affinity by molecular docking.
University of Karachi
Schiff bases of 3-formylchromone as thymidine phosphorylase inhibitors.
University of Karachi
Biotransformation of (-)-ambrox by cell suspension cultures of Actinidia deliciosa.
University of Karachi
Synthesis, in vitro β-glucuronidase inhibitory potential and molecular docking studies of quinolines.
University of Karachi
Pyridone derivative, pharmaceutical containing the same and methods of use thereof
Kaken Pharmaceutical
Synthesis, molecular docking, and biological evaluation of some novel hydrazones and pyrazole derivatives as anti-inflammatory agents.
Cairo University
Disubstituted octahydropyrrolo[3,4-c]pyrroles as orexin receptor modulators
Janssen Pharmaceutica
PIF-pocket as a target for C. albicans Pkh selective inhibitors.
Universit£Tsklinikum Frankfurt
Identification and Characterization of a New Chemotype of Noncovalent SENP Inhibitors.
Beckman Research Institute of The City of Hope
Non-amidic linkers with branched termini as CGRP receptor antagonists
Merck Sharp & Dohme
S33084, a novel, potent, selective, and competitive antagonist at dopamine D(3)-receptors: I. Receptorial, electrophysiological and neurochemical profile compared with GR218,231 and L741,626.
Centre De Recherches De Croissy
Behaviroal, pharmacological, and molecular characterization of an amphibian cannabinoid receptor.
Oregon State University
Characterization and function of the bovine kidney epithelial angiotensin receptor subtype 4 using angiotensin IV and divalinal angiotensin IV as receptor ligands.
Washington State University
Nonpeptide endothelin receptor antagonists. XI. Pharmacological characterization of SB 234551, a high-affinity and selective nonpeptide ETA receptor antagonist.
Smithkline Beecham Pharmaceuticals
Novel benzodioxopiperazines acting as antagonists at postsynaptic 5-HT1A receptors and as agonists at 5-HT1A autoreceptors: a comparative pharmacological characterization with proposed 5-HT1A antagonists.
Institut De Recherches Servier
7-Chloro-5-hydroxy-1-[2-methyl-4-(2-methylbenzoyl-amino)benzoyl ]-2,3,4,5-tetrahydro-1H-1-benzazepine (OPC-41061): a potent, orally active nonpeptide arginine vasopressin V2 receptor antagonist.
Otsuka Pharmaceutical