BindingDB

The first public molecular recognition database, BindingDB supports research, education and practice in drug discovery, pharmacology and related fields.

BindingDB contains 3.1M data for 1.3M Compounds and 9.6K Targets. Of those, 1.5M data for 698K Compounds and 4.7K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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To help with training and testing AI and other models, BindingDB downloads and search results now provide the publication date and BindingDB curation date of each measurement.

17 articles for thisTarget

The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery and early clinical development of 2-{6-[2-(3,5-dichloro-4-pyridyl)acetyl]-2,3-dimethoxyphenoxy}-N-propylacetamide (LEO 29102), a soft-drug inhibitor of phosphodiesterase 4 for topical treatment of atopic dermatitis.EBI
Leo Pharma
Melanin concentrating hormone receptor 1 (MCHR1) antagonists-Still a viable approach for obesity treatment?EBI
Leo Pharma
Synthesis and structure-activity relationship of aminobenzophenones. A novel class of p38 MAP kinase inhibitors with high antiinflammatory activity.EBI
Leo Pharma
Indolin-2-ones with high in vivo efficacy in a model for multiple sclerosis.EBI
Leo Pharma
Topical 'dual-soft' glucocorticoid receptor agonist for dermatology.EBI
Leo Pharma
Fragment-Based Discovery of 6-Arylindazole JAK Inhibitors.EBI
Leo Pharma
Synthesis, biological evaluation and SAR of 3-benzoates of ingenol for treatment of actinic keratosis and non-melanoma skin cancer.EBI
Leo Pharma
Syntheses, biological evaluation and SAR of ingenol mebutate analogues for treatment of actinic keratosis and non-melanoma skin cancer.EBI
Leo Pharma
Pyrazine compounds and uses thereofBDB
TBA
Tricyclic compounds useful to treat orthomyxovirus infectionsBDB
Novartis
Substituted indazoles, methods for the production thereof, pharmaceutical preparations that contain said new substituted indazoles, and use of said new substituted indazoles to produce drugsBDB
Bayer Pharma Aktiengesellschaft
Glutamine transport inhibitors and methods for treating cancerBDB
Vanderbilt University
Heteroaromatic carboxamide derivatives as plasma kallikrein inhibitorsBDB
Boehringer Ingelheim International
Substituted 1,2,3,4-tetrahydrobenzo[C][2,7] naphthyridines and derivatives thereof as kinase inhibitorsBDB
Allergan
Dimethyl-benzoic acid compoundsBDB
Eli Lilly
Design of potent, orally effective, nonpeptidal antagonists of the peptide hormone cholecystokinin.BDB
Merck Sharp & Dohme Research Laboratories
Sterol 14alpha-demethylase as a potential target for antitrypanosomal therapy: enzyme inhibition and parasite cell growth.BDB
Vanderbilt University