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16 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of a novel A2B adenosine receptor antagonist as a clinical candidate for chronic inflammatory airway diseases.EBI
Cv Therapeutics
2-Pyrazolyl-N(6)-substituted adenosine derivatives as high affinity and selective adenosine A(3) receptor agonists.EBI
Cv Therapeutics
Structure-affinity relationships of 5'-aromatic ethers and 5'-aromatic sulfides as partial A1 adenosine agonists, potential supraventricular anti-arrhythmic agents.EBI
Cv Therapeutics
Orally bioavailable, liver-selective stearoyl-CoA desaturase (SCD) inhibitors.EBI
Cv Therapeutics
Novel, potent, selective, and metabolically stable stearoyl-CoA desaturase (SCD) inhibitors.EBI
Cv Therapeutics
Selective, high affinity A(2B) adenosine receptor antagonists: N-1 monosubstituted 8-(pyrazol-4-yl)xanthines.EBI
Cv Therapeutics
N6-Cycloalkyl-2-substituted adenosine derivatives as selective, high affinity adenosine A1 receptor agonists.EBI
Cv Therapeutics
Novel 1,3-disubstituted 8-(1-benzyl-1H-pyrazol-4-yl) xanthines: high affinity and selective A2B adenosine receptor antagonists.EBI
Cv Therapeutics
Novel 1,3-dipropyl-8-(1-heteroarylmethyl-1H-pyrazol-4-yl)-xanthine derivatives as high affinity and selective A2B adenosine receptor antagonists.EBI
Cv Therapeutics
The discovery of a selective, high affinity A(2B) adenosine receptor antagonist for the potential treatment of asthma.EBI
Cv Therapeutics
CVT-4325: a potent fatty acid oxidation inhibitor with favorable oral bioavailability.EBI
Cv Therapeutics
New fatty acid oxidation inhibitors with increased potency lacking adverse metabolic and electrophysiological properties.EBI
Cv Therapeutics
Affinity and intrinsic efficacy (IE) of 5'-carbamoyl adenosine analogues for the A1 adenosine receptor--efforts towards the discovery of a chronic ventricular rate control agent for the treatment of atrial fibrillation (AF).EBI
Cv Therapeutics
Structure-affinity relationships of the affinity of 2-pyrazolyl adenosine analogues for the adenosine A2A receptor.EBI
Cv Therapeutics
Selective inhibition of the chymotrypsin-like activity of the 20S proteasome by 5-methoxy-1-indanone dipeptide benzamides.EBI
Cv Therapeutics
Synthesis and biological evaluation of the enantiomers of the potent and selective A1-adenosine antagonist 1,3-dipropyl-8-[2-(5,6-epoxynorbonyl)]-xanthine.EBI
Cv Therapeutics