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BindingDB contains 3.2M data for 1.4M Compounds and 11.4K Targets. Of those, 1.6M data for 748K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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10 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Structure-Based Design of an in Vivo Active Selective BRD9 Inhibitor.EBI
Boehringer Ingelheim Rcv
Detailed structure-activity relationship of indolecarboxamides as H4 receptor ligands.EBI
Boehringer Ingelheim Rcv
One-Pot Synthesis of Cereblon Proteolysis Targeting Chimeras via Photoinduced C(spEBI
Boehringer Ingelheim Rcv
Fragment Optimization of Reversible Binding to the Switch II Pocket on KRAS Leads to a Potent, In Vivo Active KRASEBI
Boehringer Ingelheim Rcv
One Atom Makes All the Difference: Getting a Foot in the Door between SOS1 and KRAS.EBI
Boehringer Ingelheim Rcv
Highly Selective PTK2 Proteolysis Targeting Chimeras to Probe Focal Adhesion Kinase Scaffolding Functions.EBI
Boehringer Ingelheim Rcv
Intracellular Trapping of the Selective Phosphoglycerate Dehydrogenase (PHGDH) Inhibitor EBI
Boehringer Ingelheim Rcv
Start Selective and Rigidify: The Discovery Path toward a Next Generation of EGFR Tyrosine Kinase Inhibitors.EBI
Boehringer Ingelheim Rcv
Bispyrimidines as potent histamine H(4) receptor ligands: delineation of structure-activity relationships and detailed H(4) receptor binding mode.EBI
Boehringer Ingelheim Rcv
Discovery and Structure-Based Optimization of Benzimidazole-Derived Activators of SOS1-Mediated Nucleotide Exchange on RAS.EBI
Boehringer Ingelheim Rcv