94 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
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SMALL-MOLECULE MODULATORS OF THE ORPHAN NUCLEAR RECEPTOR TLX
Baylor College Of Medicine
MODIFIED IMIDAZOPYRIDINES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS
Merck Sharp & Dohme
Crystalline succinate salt of 6-(6-aminopyrazin-2-yl)-n-(4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)imidazo[1,2-a]pyrazin-8-amine
Kronos Bio
DACOS type NNRTIS amino acid ester derivative, preparation method thereof, pharmaceutical composition, and application thereof
Yunnan University
Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists
Bristol-Myers Squibb
Inhibitors of tryptophan dioxygenases (IDO1 and TDO) and their use in therapy
Auckland Uniservices
Spirocycle compounds and methods of making and using same
Lundbeck La Jolla Research Center
Substituted [5,6]cyclic-4(3H)-pyrimidinones as anticancer agents
Zenji Research Laboratories
Pyridine derivatives and their use in the treatment of cancer and hemoglobinopathies
Ctxt
Spiro-condensed pyrrolidine derivatives as deubiquitylating enzymes (DUB) inhibitors
Mission Therapeutics
Heterocyclylmethyl-thienouracile as antagonists of the adenosine-A2B-receptor
Bayer Pharma Aktiengesellschaft
C2-azaspiro iminothiazine dioxides as BACE inhibitors, compositions, and their use
Merck Sharp & Dohme
Synthesis and characterization of 5,7-dihydroxyflavanone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
Yanbian University College of Pharmacy
Substituted [1,2,4]triazolo[4,3-a]pyrazines as selective NK-3 receptor antagonists
Euroscreen
Design, synthesis, and urease inhibition studies of some 1,3,4-oxadiazoles and 1,2,4-triazoles derived from mandelic acid.
Quaid-I-Azam University
Structural basis for the recognition of peptide RJPXD33 by acyltransferases in lipid A biosynthesis.
University of Michigan
Design, synthesis, cyclooxygenase inhibition and biological evaluation of new 1,3,5-triaryl-4,5-dihydro-1H-pyrazole derivatives possessing amino/methanesulfonyl pharmacophore.
Beni-Suef University
Inhibition of Pax2 Transcription Activation with a Small Molecule that Targets the DNA Binding Domain.
University of Michigan
Heat Capacity Changes for Transition-State Analogue Binding and Catalysis with Human 5'-Methylthioadenosine Phosphorylase.
Albert Einstein College of Medicine
Substituted N-(3-(pyrimidin-4-yl)phenyl)acrylamide analogs as tyrosine receptor kinase BTK inhibitors
University of Utah Research Foundation
Role of the two structural domains from the periplasmic Escherichia coli histidine-binding protein HisJ.
University of Calgary
Inhibitors of Furin and other pro-protein convertases
Sanford-Burnham Medical Research Institute
3,4-dihydropyrrolo[1,2-A]pyrazine-2,8(1H)-dicarboxamide derivatives, preparation thereof and therapeutic use thereof for diseases involving casein kinase 1 epsilon and/or casein kinase 1 delta
Sanofi
Design, synthesis, and biological characterization of tamibarotene analogs as anticancer agents.
Shandong University
Novel N-allyl/propargyl tetrahydroquinolines: Synthesis via Three-component Cationic Imino Diels-Alder Reaction, Binding Prediction, and Evaluation as Cholinesterase Inhibitors.
Universidad De Talcaa
Molecular docking studies and biological evaluation of 1,3,4-thiadiazole derivatives bearing Schiff base moieties as tyrosinase inhibitors.
Shaoyang University
Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities.
Pfizer
Substituted 3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-ones as protein kinase inhibitors
Nerviano Medical Sciences
Cosmetic compositions containing substituted azole and methods for alleviating the signs of photoaged skin
The Procter & Gamble
Amino-heteroaryl 7-hydroxy-spiropiperidine indolinyl antagonists of P2Y1 receptor
Bristol-Myers Squibb
Substituted pyrido[3,2-E][1,2,4]-triazolo[4,3-A]pyrazines for the treatment of central nervous system disorders
Boehringer Ingelheim International
Solid-Supported Synthesis and 5-HT7 /5-HT1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1H)-one.
Jagiellonian University Medical College
Fused heterocyclic derivative, medicinal composition containing the same, and medicinal use thereof
Kissei Pharmaceutical
Dimethylarginine dimethylaminohydrolase inhibitors and methods of use thereof
The Leland Stanford Junior University
Pyrimidine-substituted pyrrolidine derivatives, pharmaceutical compositions and uses thereof
Boehringer Ingelheim International
Heterocyclic pyrazole compounds, method for preparing the same and use thereof
Development Center For Biotechnology