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18 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Optimization of allosteric MEK inhibitors. Part 2: Taming the sulfamide group balances compound distribution properties.EBI
Bayer Healthcare
Neutrophil elastase inhibitors for the treatment of (cardio)pulmonary diseases: Into clinical testing with pre-adaptive pharmacophores.EBI
Bayer Healthcare
Radiofluorinated derivatives of 2-(phosphonomethyl)pentanedioic acid as inhibitors of prostate specific membrane antigen (PSMA) for the imaging of prostate cancer.EBI
Bayer Healthcare
Novel tetrahydrochinoline derived CETP inhibitors.EBI
Bayer Healthcare
Pochonins A-F, new antiviral and antiparasitic resorcylic acid lactones from Pochonia chlamydosporia var. catenulata.EBI
Bayer Healthcare
Biphenyls as potent vitronectin receptor antagonists. Part 3: Squaric acid amides.EBI
Bayer Healthcare
Optimization of imidazole amide derivatives as cannabinoid-1 receptor antagonists for the treatment of obesity.EBI
Bayer Healthcare
Constrained analogs of CB-1 antagonists: 1,5,6,7-Tetrahydro-4H-pyrrolo[3,2-c]pyridine-4-one derivatives.EBI
Bayer Healthcare
Novel, selective indole-based ECE inhibitors: lead optimization via solid-phase and classical synthesis.EBI
Bayer Healthcare
Comparison of different heterocyclic scaffolds as substrate analog PDE5 inhibitors.EBI
Bayer Healthcare
Novel heterocyclic thyromimetics.EBI
Bayer Healthcare
Optimization of allosteric MEK inhibitors. Part 1: Venturing into underexplored SAR territories.EBI
Bayer Healthcare
Novel heterocyclic thyromimetics. Part 2.EBI
Bayer Healthcare
Quinolinone pyrimidines compositions as mutant-isocitrate dehydrogenase inhibitorsBDB
Forma Tm2
Benzoxazines, benzothiazines, and related compounds having NOS inhibitory activityBDB
Neuraxon
Tyrphostins IV--highly potent inhibitors of EGF receptor kinase. Structure-activity relationship study of 4-anilidoquinazolines.BDB
Hebrew University of Jerusalem