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Targets Binding with 35 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
3-phosphoinositide-dependent protein kinase 1 [48-359]
IC50:
35
1
7
2D
3D
TSV
Acetyl-CoA carboxylase 1/2
IC50:
35
1
18
2D
3D
TSV
Baculoviral IAP repeat-containing protein 5
IC50:
1
Kd:
37
5
11
2D
3D
TSV
Beta-hexosaminidase subunit alpha
Ki:
5
IC50:
38
8
8
2D
3D
TSV
Breast cancer type 1 susceptibility protein
Ki:
18
IC50:
19
Kd:
3
3
9
2D
3D
TSV
Bromodomain and PHD finger-containing protein 3
Ki:
2
IC50:
20
Kd:
17
25
8
2D
3D
TSV
Calcium and integrin-binding protein 1
IC50:
35
Kd:
2
1
9
2D
3D
TSV
Cell surface glycoprotein MUC18
IC50:
35
1
6
2D
3D
TSV
Cytochrome P450 1A1
Ki:
10
IC50:
36
3
1
2D
3D
TSV
Dipeptidyl peptidase 8/9
IC50:
77
3
25
2D
3D
TSV
DNA polymerase
IC50:
35
1
3
2D
3D
TSV
DNA topoisomerase (ATP-hydrolyzing)
IC50:
35
1
1
2D
3D
TSV
Frizzled-7
IC50:
5
Kd:
71
1
5
2D
3D
TSV
Hsp90 co-chaperone Cdc37
IC50:
30
EC50:
25
4
3
2D
3D
TSV
Kinesin heavy chain isoform 5A
IC50:
35
3
4
2D
3D
TSV
Membrane-bound transcription factor site-1 protease
Ki:
6
IC50:
29
2
5
2D
3D
TSV
NADPH oxidase 5
Ki:
17
IC50:
18
3
12
2D
3D
TSV
Non-receptor tyrosine-protein kinase TYK2 [575-869]
EC50:
37
1
4
2D
3D
TSV
Peroxisome proliferator-activated receptor alpha [169-468]
EC50:
37
1
8
2D
3D
TSV
Prostaglandin G/H synthase 2 [E165G]
IC50:
36
2
4
2D
3D
TSV
Prostaglandin-H2 D-isomerase
Ki:
7
IC50:
35
6
17
2D
3D
TSV
RuvB-like 1
IC50:
37
2
9
2D
3D
TSV
Ryanodine receptor 1 [4317-4329]
IC50:
35
1
6
2D
3D
TSV
Serine hydroxymethyltransferase, mitochondrial
IC50:
67
3
7
2D
3D
TSV
Transmembrane protease serine 2
Ki:
9
IC50:
23
EC50:
5
9
9
2D
3D
TSV
Tyrosine-protein phosphatase non-receptor type 13
Ki:
1
IC50:
44
13
12
2D
3D
TSV