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Targets Binding with 26 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
1-phosphatidylinositol 3-phosphate 5-kinase [1-2098,S696N,L932S,Q995L,T998S,S1033A,Q1183K]
IC50:
29
1
14
2D
3D
TSV
A disintegrin and metalloproteinase with thrombospondin motifs 1
Ki:
5
IC50:
22
4
7
2D
3D
TSV
Arachidonate 12-lipoxygenase, 12R-type
Ki:
2
IC50:
24
3
1
2D
3D
TSV
Bromodomain testis-specific protein [21-137]
Ki:
2
IC50:
24
Kd:
1
1
12
2D
3D
TSV
CAAX prenyl protease 2
IC50:
26
3
3
2D
3D
TSV
Calpain small subunit 1
Ki:
27
4
3
2D
3D
TSV
Carnitine O-palmitoyltransferase 2, mitochondrial
Ki:
8
IC50:
32
3
7
2D
3D
TSV
Citrate synthase, peroxisomal [1-24]
EC50:
26
2
3
2D
3D
TSV
Cytochrome P450 2C18
IC50:
26
2
7
2D
3D
TSV
DNA topoisomerase 4 subunit B
Ki:
2
IC50:
27
5
6
2D
3D
TSV
DNA-binding protein Ikaros
EC50:
28
1
9
2D
3D
TSV
Dual specificity mitogen-activated protein kinase kinase 1/RAF proto-oncogene serine/threonine-protein kinase
IC50:
26
2
6
2D
3D
TSV
Epidermal growth factor receptor [L858R,C797S]
IC50:
27
2
16
2D
3D
TSV
Fe(3+)-Zn(2+) purple acid phosphatase
Ki:
25
IC50:
6
4
3
2D
3D
TSV
Glucose-induced degradation protein 4 homolog
IC50:
25
Kd:
4
1
4
2D
3D
TSV
Histone-binding protein RBBP4/Histone-lysine N-methyltransferase EZH1/Polycomb protein EED/Polycomb protein SUZ12/Zinc finger protein AEBP2
IC50:
26
2
30
2D
3D
TSV
HLA class II histocompatibility antigen, DR beta 3 chain
IC50:
27
1
47
2D
3D
TSV
Inhibitor of nuclear factor kappa-B kinase subunit epsilon/Serine/threonine-protein kinase TBK1
IC50:
26
1
9
2D
3D
TSV
N-glycosylase/DNA lyase
IC50:
32
2
18
2D
3D
TSV
NAD-dependent protein deacetylase HST2
Ki:
8
IC50:
16
Kd:
11
2
3
2D
3D
TSV
Peptidase
IC50:
45
Kd:
5
Koff:
4
8
4
2D
3D
TSV
Phospholipase D
IC50:
42
2
2
2D
3D
TSV
Platelet-activating factor acetylhydrolase IB subunit alpha2
IC50:
35
2
13
2D
3D
TSV
Platelet-derived growth factor subunit B
Ki:
1
IC50:
24
Kd:
1
4
7
2D
3D
TSV
Poly [ADP-ribose] polymerase tankyrase-1 [1112-1317]
IC50:
26
1
5
2D
3D
TSV
Poly [ADP-ribose] polymerase tankyrase-2 [959-1164]
IC50:
26
1
5
2D
3D
TSV
Prostaglandin reductase 2
IC50:
26
EC50:
26
1
4
2D
3D
TSV
Protein arginine N-methyltransferase 7
IC50:
30
Kd:
1
12
7
2D
3D
TSV
Pyrroline-5-carboxylate reductase
Ki:
3
IC50:
52
2
1
2D
3D
TSV
Resistin
IC50:
26
1
5
2D
3D
TSV
Retinoic acid receptor RXR-alpha/Thyroid hormone receptor alpha
EC50:
27
1
9
2D
3D
TSV
Retinoic acid receptor RXR-alpha/Thyroid hormone receptor beta
EC50:
27
1
11
2D
3D
TSV
Tyrosine-protein phosphatase 1
IC50:
26
6
3
2D
3D
TSV
UDP-glucuronosyltransferase 1-6
Ki:
4
IC50:
23
6
5
2D
3D
TSV
Voltage-dependent L-type calcium channel subunit beta-1/N-type calcium channel subunit alpha-1B/calcium channel subunit alpha-2/delta-1
IC50:
27
2
18
2D
3D
TSV