Compile Data Set for Download or QSAR
Report error Found 1493 of affinity data for UniProtKB/TrEMBL: Q9Y337
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525914(CHEMBL4558285)
Affinity DataIC50: 0.316nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525895(CHEMBL4447752)
Affinity DataIC50: 0.501nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525899(CHEMBL4465265)
Affinity DataIC50: 0.794nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525904(CHEMBL4461533)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525912(CHEMBL4543039)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525918(CHEMBL4473069)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525895(CHEMBL4447752)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525917(CHEMBL4579813)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525914(CHEMBL4558285)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525899(CHEMBL4465265)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525905(CHEMBL4517343)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525912(CHEMBL4543039)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525903(CHEMBL4436048)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525917(CHEMBL4579813)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525904(CHEMBL4461533)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525897(CHEMBL4536142)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525913(CHEMBL4464120)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525905(CHEMBL4517343)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525911(CHEMBL4535907)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522475(CHEMBL4535831)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525911(CHEMBL4535907)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525901(CHEMBL4448315)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525913(CHEMBL4464120)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525918(CHEMBL4473069)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525901(CHEMBL4448315)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525897(CHEMBL4536142)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525903(CHEMBL4436048)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525900(CHEMBL4460168)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525902(CHEMBL4547455)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525900(CHEMBL4460168)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522496(CHEMBL4586700)
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522495(CHEMBL4435372)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525902(CHEMBL4547455)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522494(CHEMBL4458360)
Affinity DataIC50: 63nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM32881([3-(2-furanyl)-5-(methylthio)-1,2,4-triazol-1-yl]-...)
Affinity DataIC50: 76nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Scott L. Diamond, University of Pennsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522475(CHEMBL4535831)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522485(CHEMBL4471660)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522477(CHEMBL4576787)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522488(CHEMBL4452547)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522493(CHEMBL4530083)
Affinity DataIC50: 79nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50525920(CHEMBL4465992)
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant 6His-Q-FLAG-tagged KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM33906(SMR000378089 | 5-amino-1-[(4-methoxyphenyl)-oxomet...)
Affinity DataIC50: 84.4nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Scott L. Diamond, University of Pennsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM32765(cid_658532 | prop-2-ynyl 2-(benzotriazol-1-ylcarbo...)
Affinity DataIC50: 87.1nMAssay Description:Molecular Library Screening Center Network (MLSCN) Penn Center for Molecular Discovery (PCMD) Assay Provider: Scott L. Diamond, University of Pennsy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2011
Entry Details
PCBioAssay
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522487(CHEMBL4593503)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50154254(CHEMBL3775705)
Affinity DataIC50: 112nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50154253(CHEMBL3775377)
Affinity DataIC50: 115nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM50154252(CHEMBL3774934)
Affinity DataIC50: 122nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50522486(CHEMBL4517626)
Affinity DataIC50: 126nMAssay Description:Inhibition of recombinant 6His-Q-FLAG tagged human KLK5 expressed in baculovirus infected Sf9 insect cells using (Tos-Gly-Pro-Arg)2[R110].2TFA as sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetKallikrein-5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)
Affinity DataIC50: 130nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Universidade Federal Fluminense

Curated by ChEMBL
LigandPNGBDBM51911(3-(2-methoxyphenyl)-3-(4-methoxyphenyl)-N-[(4-prop...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
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