Compile Data Set for Download or QSAR
Report error Found 7 of affinity data for UniProtKB/TrEMBL: Q9UM81
TargetProtein-tyrosine-phosphatase(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391713(CHEMBL2146956)
Affinity DataIC50: 100nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein-tyrosine-phosphatase(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50237957(4-(2-((2,5-dioxoimidazolidin-4-ylidene)methyl)-1H-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein-tyrosine-phosphatase(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391714(CHEMBL2146957)
Affinity DataIC50: 600nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein-tyrosine-phosphatase(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391715(CHEMBL2146960)
Affinity DataIC50: 700nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein-tyrosine-phosphatase(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391711(CHEMBL2146958)
Affinity DataIC50: 900nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein-tyrosine-phosphatase(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387974(CHEMBL2057830)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein-tyrosine-phosphatase(Human)
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391712(CHEMBL2146959)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed