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Report error Found 35 of affinity data for UniProtKB/TrEMBL: Q9JIM1
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457379(CHEMBL4211925)
Affinity DataIC50: 14nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457390(CHEMBL4208680)
Affinity DataIC50: 17nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457381(CHEMBL4211194)
Affinity DataIC50: 18nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457387(CHEMBL4215413)
Affinity DataIC50: 24nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457386(CHEMBL4212967)
Affinity DataIC50: 26nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409054(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...)
Affinity DataIC50: 27nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457385(CHEMBL4207561)
Affinity DataIC50: 27nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409053(6-(5-Fluoro-6-methylpyridin-3-yl)-3,3-dimethyl-1-(...)
Affinity DataIC50: 27nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457378(CHEMBL4203736)
Affinity DataIC50: 31nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409033(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...)
Affinity DataIC50: 32.1nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409050(1-(6-Cyclopropyl-5-(methylsulfonyl)pyridin-3-yl)-3...)
Affinity DataIC50: 38.5nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457384(CHEMBL4210157)
Affinity DataIC50: 39nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409044(1-(5-(Cyclopropylsulfonyl)pyridin-3-yl)-3,3-dimeth...)
Affinity DataIC50: 40nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409034(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(6-(meth...)
Affinity DataIC50: 40.1nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409037(5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...)
Affinity DataIC50: 44.9nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457376(CHEMBL4213616)
Affinity DataIC50: 52nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457377(CHEMBL4205790)
Affinity DataIC50: 57nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409049(5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...)
Affinity DataIC50: 71.7nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409048(5-(3,3-dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...)
Affinity DataIC50: 79.3nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457388(CHEMBL4217494)
Affinity DataIC50: 97nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409035(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(3-(meth...)
Affinity DataIC50: 106nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409046(5-(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-2-oxoin...)
Affinity DataIC50: 128nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409043(1-(5-(Isopropylsulfonyl)pyridin-3-yl)-3,3-dimethyl...)
Affinity DataIC50: 135nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409055(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...)
Affinity DataIC50: 157nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409047(1-(5-(Azetidin-1-ylsulfonyl)pyridin-3-yl)-3,3-dime...)
Affinity DataIC50: 169nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409031(1-(Benzo[b]thiophen-6-yl)-3,3-dimethyl-6-(2-methyl...)
Affinity DataIC50: 189nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409051(3,3-Dimethyl-6-(2-methyl-1-oxidopyrimidin-1-ium-5-...)
Affinity DataIC50: 218nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409045(3,3-Dimethyl-6-(2-methylpyrimidin-5-yl)-1-(5-(meth...)
Affinity DataIC50: 218nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409056(6'-(2-Methylpyrimidin-5-yl)-1'-(5-(methylsulfonyl)...)
Affinity DataIC50: 230nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457380(CHEMBL4206265)
Affinity DataIC50: 244nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457383(CHEMBL4216732)
Affinity DataIC50: 253nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409052(3,3-Dimethyl-6-(5-methylpyridin-3-yl)-1-(5-(methyl...)
Affinity DataIC50: 313nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent

TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457382(CHEMBL4213885)
Affinity DataIC50: 321nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM50457389(CHEMBL4212469)
Affinity DataIC50: 838nMAssay Description:Inhibition of mouse ENT1 expressed in mammalian cells assessed as reduction in [2,8-H]adenosine uptake by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Mouse)
Dart Neuroscience

Curated by ChEMBL
LigandPNGBDBM409032(1-(Benzo[b]thiophen-4-yl)-3,3-dimethyl-6-(2-methyl...)
Affinity DataIC50: 844nMAssay Description:To measure adenosine transport activity of ENT-1 mammalian cells, stable cells expressing the mouse ENT-1 transporter were plated on day 1 in 96-well...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2020
Entry Details
Go to US Patent