Compile Data Set for Download or QSAR
Report error Found 167 of affinity data for UniProtKB/TrEMBL: Q9HBW0
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148349((3-Octadec-9-enoylamino-propionyl)-phosphonothioic...)
Affinity DataEC50:  108nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  6.80nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148350([3-((Z)-Octadec-9-enoylamino)-thiopropionyl]-phosp...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148351([3-((Z)-Octadec-9-enoylamino)-propionyl]-phosphoni...)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148352([1-Hydroxy-3-((Z)-octadec-9-enoylamino)-propyl]-ph...)
Affinity DataEC50:  2.07E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50074700(Phosphoric acid mono-[2-((Z)-octadec-9-enoylamino)...)
Affinity DataEC50:  30nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148354([1-Fluoro-3-((Z)-octadec-9-enoylamino)-propyl]-pho...)
Affinity DataEC50:  1.96E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148353((1-Hydroxy-3-octadec-9-enoylamino-1-phosphono-prop...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148355([3-((Z)-Octadec-9-enoylamino)-propyl]-phosphonic a...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 2 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056342(CHEMBL3322509)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056343(CHEMBL3322513)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056344(CHEMBL3322514)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056345(CHEMBL3322500)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056346(CHEMBL3322501)
Affinity DataEC50:  2.16E+3nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056347(CHEMBL3322502)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056348(CHEMBL3322503)
Affinity DataEC50:  1.42E+3nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056349(CHEMBL3322507)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50056350(CHEMBL3322508)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human LPA2 expressed in LPA1xLPA2 double knockout mouse MEF cells by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/31/2016
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170852(Thiophosphoric acid (E)-tetradec-9-enyl ester | CH...)
Affinity DataEC50:  480nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170850(Phosphoric acid monodecyl ester | CHEMBL361255)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170855(Thiophosphoric acid dec-9-enyl ester | CHEMBL36393...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170857(Thiophosphoric acid decyl ester | CHEMBL187795)
Affinity DataEC50:  4.57E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170854(Phosphoric acid monododecyl ester | CHEMBL187711)
Affinity DataEC50:  3.10E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170860(Thiophosphoric acid dodecyl ester | CHEMBL191365)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170858(Phosphoric acid mono-((E)-dodec-9-enyl) ester | CH...)
Affinity DataEC50:  717nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170856(Phosphoric acid mono-((E)-dec-4-enyl) ester | CHEM...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170844(Thiophosphoric acid (E)-octadec-9-enyl ester | CHE...)
Affinity DataEC50:  244nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170843(Phosphoric acid mono-((E)-tetradec-9-enyl) ester |...)
Affinity DataEC50:  397nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170849(Thiophosphoric acid tetradecyl ester | CHEMBL18929...)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170863(Phosphoric acid monodec-9-enyl ester | CHEMBL36377...)
Affinity DataEC50:  3.80E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170847(Thiophosphoric acid (E)-dodec-9-enyl ester | CHEMB...)
Affinity DataEC50:  677nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170851(Phosphoric acid mono-((E)-tetradec-11-enyl) ester ...)
Affinity DataEC50:  4.10E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50176394(octanoic acid (R)-2-octanoyloxy-3-thiophosphonooxy...)
Affinity DataEC50:  6.33E+3nMAssay Description:Activity at LPA2 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50176390((R)-O-2,3-bis(octyloxy)propyl O,O-dihydrogen phosp...)
Affinity DataEC50:  5.72E+3nMAssay Description:Activity at LPA2 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50176399(octanoic acid (S)-2-octanoyloxy-3-thiophosphonooxy...)
Affinity DataEC50:  7.17E+3nMAssay Description:Activity at LPA2 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177335(potassium O-((2R,4R)-2-(heptadec-9-enyl)-1,3-dioxo...)
Affinity DataEC50:  1.09E+3nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177336(potassium (2-(heptadec-9-enyl)-1,3-dioxolan-4-yl)m...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177328(potassium O-((2S,4R)-2-(heptadec-9-enyl)-1,3-dioxo...)
Affinity DataEC50:  1.30E+3nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177338(potassium (2-(heptadeca-9,12,15-trienyl)-1,3-dioxo...)
Affinity DataEC50:  1.71E+3nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177340(potassium ((2R,4S)-2-(heptadec-9-enyl)-1,3-dioxola...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177339(potassium ((2R,4R)-2-(heptadec-9-enyl)-1,3-dioxola...)
Affinity DataEC50:  1.71E+3nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177330(potassium O-((2S,4S)-2-(heptadec-9-enyl)-1,3-dioxo...)
Affinity DataEC50:  1.32E+3nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177333(potassium O-((2R,4S)-2-(heptadec-9-enyl)-1,3-dioxo...)
Affinity DataEC50:  1.54E+3nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177341(potassium ((2S,4R)-2-(heptadec-9-enyl)-1,3-dioxola...)
Affinity DataEC50:  1.17E+3nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50177332(potassium O-(2-(heptadec-9-enyl)-1,3-dioxolan-4-yl...)
Affinity DataEC50:  1.17E+3nMAssay Description:Activity at LPA2 receptor in RH7777 rat hepatoma cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50193516(1,1-difluoro-3(S)-hydroxyl-4-oleoyloxylbutane 1,3-...)
Affinity DataEC50: >9.46E+3nMAssay Description:Activity at human LPA2 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50271700(4-(4-(ethoxycarbonyl)styryl)benzenesulfonic acid |...)
Affinity DataEC50: >1.14E+4nMAssay Description:Agonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human LPA2 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 2(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50381022(CHEMBL2017139)
Affinity DataEC50:  161nMAssay Description:Agonist activity at human LPA2 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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