Compile Data Set for Download or QSAR
Report error Found 2607 of affinity data for UniProtKB/TrEMBL: Q9H3N8
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataEC50:  25.1nMAssay Description:Agonist activity at human histamine H4 receptor expressed in HEK293 cells assessed by forskolin induced cAMP response element activation by luciferas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataEC50:  79.4nMAssay Description:Inverse agonist activity at human histamine H4 receptor expressed in HEK293 cells assessed by forskolin induced cAMP response element activation by l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50418058(CHEMBL1688946)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human histamine H4 receptor expressed in HEK293 cells assessed by forskolin induced cAMP response element activation by luciferas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50418059(CHEMBL1688969)
Affinity DataEC50:  158nMAssay Description:Agonist activity at human histamine H4 receptor expressed in HEK293 cells assessed by forskolin induced cAMP response element activation by luciferas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM22543(2-[4-(1H-imidazol-4-ylmethyl)phenyl]-4,4-dimethyl-...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Ligand displacement assays were performed on CHO cells membranes expressing hH4R. Retained radioactivity was determined by liquid scintillation count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2008
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127604(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127608(2-[2-(1H-Imidazol-4-yl)-cyclopropyl]-ethylamine | ...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127605(VUF-5297 | (1S,2S)-2-(1H-Imidazol-4-yl)-cyclopropy...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127607(VUF-5296 | 2-(1H-Imidazol-4-yl)-cyclopropylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127601(2-(1H-Imidazol-4-yl)-cyclopropylamine | CHEMBL5938...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127602(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127609(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127603(C-[2-(1H-Imidazol-4-yl)-cyclopropyl]-methylamine |...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127610((1S,2S)-2-(2-aminoethyl)-1-(1H-imidazol-4-yl)cyclo...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50127606(2-(1H-Imidazol-4-yl)-cyclopropylamine | CHEMBL2940...)
Affinity DataEC50: >0.000100nMAssay Description:Inhibition of human Histamine H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006739(CHEMBL3236552)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006742(CHEMBL3236553)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006743(CHEMBL3236554)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006744(CHEMBL3236555)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006745(CHEMBL3236556)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006746(CHEMBL3236557)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006747(CHEMBL3236558)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006749(CHEMBL3236560)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006750(CHEMBL3236561)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006751(CHEMBL3236562)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006753(CHEMBL3236564)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006754(CHEMBL3236565)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006755(CHEMBL3233048)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006758(CHEMBL3236568)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006759(CHEMBL3236569)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006760(CHEMBL3236570)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006761(CHEMBL3236571)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006762(CHEMBL3236572)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006764(CHEMBL3236574)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006765(CHEMBL3236575)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006766(CHEMBL3236576)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006767(CHEMBL3236577)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006768(CHEMBL3236578)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006769(CHEMBL3236579)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50006772(CHEMBL3236582)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human H4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413503(UR-PI141 | CHEMBL514641)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413504(CHEMBL474449)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413502(UR-PI104 | CHEMBL474447)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50377986(UR-AK24 | CHEMBL483406)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413506(UR-PI147 | CHEMBL474617)
Affinity DataEC50:  151nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413505(CHEMBL515428)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413500(UR-PI287 | CHEMBL471724)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50413501(SK&F-91486 | SK-91486 | CHEMBL325327)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at human H4 receptor expressed in insect Sf9 cells co-expressing RGS19 fusion protein and Gialpha2, Gbeta1gamma2 assessed as gamma[3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Displayed 1 to 50 (of 2607 total ) | Next | Last >>
Jump to: