Compile Data Set for Download or QSAR
Report error Found 39 for UniProtKB: Q9ERZ4
LigandPNGBDBM83449(cid_9795678 | PHENCYCLIDINE | SMR001338811 | Phenc...)
Affinity DataKd:  9.10E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor was determined by using [3H]4NMPB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50028052(Allyl-ethyl-(1-phenyl-cyclohexyl)-amine | CHEMBL23...)
Affinity DataKd:  1.40E+4nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor was determined by using [3H]4NMPB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50028051(Diallyl-(1-phenyl-cyclohexyl)-amine | CHEMBL23626)
Affinity DataKd:  2.50E+4nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor was determined by using [3H]4NMPB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50028053(Allyl-methyl-(1-phenyl-cyclohexyl)-amine | CHEMBL2...)
Affinity DataKd:  1.50E+4nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor was determined by using [3H]4NMPB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50028054(Allyl-(1-phenyl-cyclohexyl)-amine | CHEMBL281855)
Affinity DataKd:  7.00E+4nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor was determined by using [3H]4NMPB as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005492(CHEMBL418712 | {5-[9-(5-Dimethylaminomethyl-furan-...)
Affinity DataIC50: 400nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005493(CHEMBL12858 | N-((5-Ethylsulfanylmethyl-furan-2-yl...)
Affinity DataIC50: 470nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005504(CHEMBL13206 | N-((5-Ethylsulfanylmethyl-furan-2-yl...)
Affinity DataIC50: 500nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005495(CHEMBL13166 | {5-[5-(5-Dimethylaminomethyl-furan-2...)
Affinity DataIC50: 520nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005494(CHEMBL418714 | {5-[8-(5-Dimethylaminomethyl-furan-...)
Affinity DataIC50: 540nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005502(CHEMBL12472 | {5-[4-(5-Dimethylaminomethyl-furan-2...)
Affinity DataIC50: 550nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005509(CHEMBL268499 | {5-[6-(5-Dimethylaminomethyl-furan-...)
Affinity DataIC50: 580nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005500(CHEMBL13122 | N,N'-Bis-[2-(5-dimethylaminomethyl-f...)
Affinity DataIC50: 590nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005496(CHEMBL13426 | {5-[7-(5-Dimethylaminomethyl-furan-2...)
Affinity DataIC50: 710nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005503(CHEMBL13308 | {5-[2-(5-Dimethylaminomethyl-furan-2...)
Affinity DataIC50: 1.40E+3nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005501(CHEMBL275537 | {5-[3-(5-Dimethylaminomethyl-furan-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005498(CHEMBL12781 | {5-[4'-(5-Dimethylaminomethyl-furan-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 2.10E+3nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50005497(CHEMBL12937 | {5-[4-(5-Dimethylaminomethyl-furan-2...)
Affinity DataIC50: 2.20E+3nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
LigandPNGBDBM50020529(CHEMBL34000 | 2-(Hydroxyimino-methyl)-3-methyl-1-(...)
Affinity DataIC50: 2.20E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic acetylcholine receptor in mouse brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
LigandPNGBDBM50020515(CHEMBL33332 | 2-(Hydroxyimino-methyl)-3-methyl-1-(...)
Affinity DataIC50: 3.50E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic acetylcholine receptor in mouse brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
LigandPNGBDBM50020521(CHEMBL32585 | 2-(Hydroxyimino-methyl)-3-methyl-1-(...)
Affinity DataIC50: 8.00E+4nMAssay Description:Compound was tested for the binding affinity towards muscarinic acetylcholine receptor in mouse brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 1.60E+5nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]methylscopolamine binding to Muscarinic acetylcholine receptor M2 of mouse cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
LigandPNGBDBM50020522(1-(((4-carbamoylpyridinium-1-yl)methoxy)methyl)-2-...)
Affinity DataIC50: 1.60E+5nMAssay Description:Compound was tested for the binding affinity towards muscarinic acetylcholine receptor in mouse brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
LigandPNGBDBM50011780(Pralidoxine chloride | PRALIDOXIME | CHEMBL748 | 2...)
Affinity DataIC50: 1.70E+5nMAssay Description:Compound was tested for the binding affinity towards muscarinic acetylcholine receptor in mouse brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
LigandPNGBDBM50020514(CHEMBL289890 | 2-(Hydroxyimino-methyl)-1-methoxyme...)
Affinity DataIC50: 1.00E+6nMAssay Description:Compound was tested for the binding affinity towards muscarinic acetylcholine receptor in mouse brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.350nMAssay Description:Ability to displace [3H]oxotremorine ([3H]-OXO-M) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKi:  0.700nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataKi:  1.70nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  8nMAssay Description:Ability to displace [3H]oxotremorine ([3H]OXO-M) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataKi:  220nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004664(CHEMBL107892 | N-[2-(5-Dimethylaminomethyl-furan-2...)
Affinity DataKi:  460nMAssay Description:Ability to displace [3H]oxotremorine ([3H]-OXO-M) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004661(CHEMBL316973 | [2-(5-Dimethylaminomethyl-furan-2-y...)
Affinity DataKi:  870nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004652(CHEMBL321605 | [2-(5-Dimethylaminomethyl-furan-2-y...)
Affinity DataKi:  1.10E+3nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataKi:  1.50E+3nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004664(CHEMBL107892 | N-[2-(5-Dimethylaminomethyl-furan-2...)
Affinity DataKi:  9.50E+3nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004652(CHEMBL321605 | [2-(5-Dimethylaminomethyl-furan-2-y...)
Affinity DataKi:  1.20E+4nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004661(CHEMBL316973 | [2-(5-Dimethylaminomethyl-furan-2-y...)
Affinity DataKi:  1.20E+4nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Mouse)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  6.60E+4nMAssay Description:Ability to displace [3H]methylscopolamine ([3H]NMS) from mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed