Compile Data Set for Download or QSAR
Report error Found 394 of affinity data for UniProtKB/TrEMBL: Q9BYT3
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM21079(1-[4-(3-azanyl-1H-indazol-4-yl)phenyl]-3-(2-fluora...)
Affinity DataKd:  3.80E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31085(cid_11409972 | 1-[4-[(4-ethylpiperazin-1-yl)methyl...)
Affinity DataKd:  1.20E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-etho...)
Affinity DataKd:  4.50E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31099(CHEMBL45741 | Flavopiridol | cid_24867231 | 2-(2-c...)
Affinity DataKd:  1.70E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM17055((9S)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydr...)
Affinity DataKd:  3.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd:  130nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataKd:  2.40E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705 | US2024...)
Affinity DataKd:  1.80nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  17nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM21(VANDETANIB | N-(4-bromo-2-fluorophenyl)-6-methoxy-...)
Affinity DataKd:  1.40E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67642(5-(4-Hydroxy-3-methoxy-benzylidene)-2-(2-methoxy-p...)
Affinity DataEC50:  4.00E+3nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67643(SMR000513437 | MLS001209287 | 4-[(3-Mercapto-5-phe...)
Affinity DataEC50:  2.58E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67644(N2-(4-ethoxyphenyl)quinazoline-2,4-diamine;hydroch...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67645(The compound has not trivial name. | SMR000518462 ...)
Affinity DataEC50:  2.27E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67646(MLS001206211 | [(Z)-[azanyl(pyridin-2-yl)methylide...)
Affinity DataEC50:  3.22E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67647(SMR000523783 | cid_956331 | Benzothiazol-2-yl-(3,4...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67648(The compound has not trivial name. | 2-[[3-[(2-car...)
Affinity DataEC50:  5.96E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67649(MLS001212262 | cid_5408200 | N-methyl-N-[4-[[(Z)-(...)
Affinity DataEC50:  3.76E+3nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67650(4-[(2-Hydroxy-naphthalen-1-ylmethylene)-amino]-3-m...)
Affinity DataEC50:  2.27E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67651(SMR000504332 | 3-(6-azanyl-5-nitro-4-phenyl-pyridi...)
Affinity DataEC50: <100nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM59052((5Z)-2-azanyl-5-[(3-methoxy-4-oxidanyl-phenyl)meth...)
Affinity DataEC50:  936nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67652(cid_3097937 | SMR000513323 | 9-Hydroxyimino-9H-flu...)
Affinity DataEC50:  4.91E+3nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM60883(2-Chloro-5-[5-(2,3-dibromo-4-hydroxy-5-methoxy-ben...)
Affinity DataEC50:  1.59E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67653((4E)-4-[[(3-cyclohexyl-5-sulfanylidene-1H-1,2,4-tr...)
Affinity DataEC50:  2.20E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67654(SMR000539302 | MLS001163883 | (6E)-6-[4-(4-methyl-...)
Affinity DataEC50:  4.28E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67655(decyl 2-[2-[(4-chloranylphenoxy)methyl]-3-methyl-b...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM58367(MLS001165405 | [(3Z)-3-(2-chlorothioxanthen-9-ylid...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM51912([(3Z)-3-(2-chloro-9-thioxanthenylidene)propyl]-dec...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67656(N-[5,6-bis(4-methoxyphenyl)furo[2,3-d]pyrimidin-4-...)
Affinity DataEC50:  3.36E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67657(MLS001165184 | cid_6083642 | (6E)-6-[4-[4-(2-hydro...)
Affinity DataEC50:  2.31E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67658(2-[2-(1-methyl-2-pyrrolidinyl)ethylamino]-9-thioxa...)
Affinity DataEC50:  1.66E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67659(cid_24747911 | 2-(3-morpholin-4-ylpropylamino)thio...)
Affinity DataEC50:  1.68E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67660((5Z)-5-[(3-ethoxy-4-hydroxyphenyl)methylidene]-2-(...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67661(The compound has not trivial name. | MLS001210481 ...)
Affinity DataEC50:  2.18E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67662((E)-3-(dimethylamino)-1-[3-(4-methoxyphenyl)-2,1-b...)
Affinity DataEC50:  5.29E+3nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67663(cid_1485416 | SMR000550248 | N-methyl-N'-[3-(2...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67664(MLS001165915 | cid_5902388 | (E)-3-(dimethylamino)...)
Affinity DataEC50:  1.20E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67665((E)-3-(dimethylamino)-1-[3-(3-fluorophenyl)-2,1-be...)
Affinity DataEC50:  1.87E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67666(SMR000549693 | MLS001166481 | cid_1483761 | (E)-3-...)
Affinity DataEC50:  1.59E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67667(MLS001214182 | N-(3-oxidanylpropyl)-1-phenyl-9H-py...)
Affinity DataEC50:  2.34E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67668(cid_6097961 | CHEMBL1487936 | (6E)-6-[4-[(4-hydrox...)
Affinity DataEC50:  2.43E+3nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67669(cid_5338745 | N'-[(4-methoxybenzoyl)oxy]benzen...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67670(MLS001182271 | SMR000568075 | cid_2743674 | N-[[2,...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67671(SMR000590970 | MLS001170902 | 2-[4-[(E)-3-[2-[(4-m...)
Affinity DataEC50:  1.86E+3nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67672(MLS001173801 | 2-chloro-5-[[(Z)-(2-oxo-1-naphthale...)
Affinity DataEC50:  3.23E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM32069((11S)-11-methyl-15,17-bis(oxidanyl)-12-oxabicyclo[...)
Affinity DataEC50:  4.46E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM7238(cid_5289419 | 3-(3H-Imidazol-4-ylmethylene)-5-meth...)
Affinity DataEC50:  7.73E+3nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67673(cid_20854282 | 6-{[(2-fluorophenyl)amino]sulfonyl}...)
Affinity DataEC50: >1.20E+5nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67674(4-[[6-[(4-carboxyphenyl)carbamoyl]pyridin-2-yl]car...)
Affinity DataEC50:  2.83E+4nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
TargetSerine/threonine-protein kinase 33(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM67675(N-[2-(3-oxo-4H-quinoxalin-2-yl)phenyl]-2-thiophene...)
Affinity DataEC50:  2.10E+3nMAssay Description:Keywords: STK33 Kinase, Non-ATP Competitive Inhibitor Assay Overview: Purified STK33 Kinase is preincubated with potential inhibitors and allowed to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2011
Entry Details
PCBioAssay
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