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Report error Found 636 of affinity data for UniProtKB/TrEMBL: Q99873
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50206427(AMI-1 | 7,7'-carbonylbis(azanediyl)bis(4-hydroxyna...)
Affinity DataKd:  810nMAssay Description:Binding affinity to human recombinant GST-PRMT1 expressed Escherichia coli BL21 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  3.69E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataKd:  4.24E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50590375(CHEMBL5187396)
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM588052((2R)-7-chloro-2-[trans-4-(dimethylamino)cyclohexyl...)
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636218(CHEMBL5559689)
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636218(CHEMBL5559689)
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50648689(CHEMBL5612531)
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636218(CHEMBL5559689)
Affinity DataIC50: 3.10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636218(CHEMBL5559689)
Affinity DataIC50: 3.20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095354(CHEMBL3589030)
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095432(CHEMBL3589026)
Affinity DataIC50: 4nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM178103(MS023 (Compound 3) | N1-((4-(4-isopropoxyphenyl)-1...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human PRMT1 assessed as inhibition of methylation activity using biotin-labeled peptide as substrate and [3H]-SAM by scintillation prox...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2018
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM178103(MS023 (Compound 3) | N1-((4-(4-isopropoxyphenyl)-1...)
Affinity DataIC50: 4nMAssay Description:Inhibition of PRMT1 (unknown origin) using biotinylated histone H4 (1 to 24 residues) as substrate in presence of [3H]SAM by scintillation proximity ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM178103(MS023 (Compound 3) | N1-((4-(4-isopropoxyphenyl)-1...)
Affinity DataIC50: 4nMAssay Description:Inhibition of PRMT1 (unknown origin) by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636201(CHEMBL5517922)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636202(CHEMBL5527874)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095353(CHEMBL3589031)
Affinity DataIC50: 5nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095356(CHEMBL3589028)
Affinity DataIC50: 5nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636206(CHEMBL5565736)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50651366(CHEMBL5633975)
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50637545(CHEMBL5532081)
Affinity DataIC50: 5.90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095355(CHEMBL3589029)
Affinity DataIC50: 7nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095357(CHEMBL3589027)
Affinity DataIC50: 7nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095348(CHEMBL3589036)
Affinity DataIC50: 8nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636200(CHEMBL5542306)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636204(CHEMBL5532462)
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636218(CHEMBL5559689)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50643941(CHEMBL5567635)
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50643940(CHEMBL5566241)
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095351(CHEMBL3589033)
Affinity DataIC50: 13nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095433(CHEMBL3589913)
Affinity DataIC50: 13nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095347(CHEMBL3589037)
Affinity DataIC50: 14nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095352(CHEMBL3589032)
Affinity DataIC50: 14nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636212(CHEMBL5560201)
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636210(CHEMBL5557453)
Affinity DataIC50: 15nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095442(CHEMBL3589038)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636203(CHEMBL5561358)
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50636205(CHEMBL5558900)
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50648690(CHEMBL5613916)
Affinity DataIC50: 17nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095434(CHEMBL3589912)
Affinity DataIC50: 18nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM502122(US11028083, Example 91)
Affinity DataIC50: 22nMAssay Description:This enzymatic assay was performed in a 384 well, white, low volume plate (PerkinElmer, Catalog 6008289) with assay buffer consisting of 50 mM Hepes ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM502138(US11028083, Example 100b)
Affinity DataIC50: 22nMAssay Description:This enzymatic assay was performed in a 384 well, white, low volume plate (PerkinElmer, Catalog 6008289) with assay buffer consisting of 50 mM Hepes ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM502103(US11028083, Example 80b | US11028083, Example 79b)
Affinity DataIC50: 24nMAssay Description:This enzymatic assay was performed in a 384 well, white, low volume plate (PerkinElmer, Catalog 6008289) with assay buffer consisting of 50 mM Hepes ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM502116(US11028083, Example 87b)
Affinity DataIC50: 24nMAssay Description:This enzymatic assay was performed in a 384 well, white, low volume plate (PerkinElmer, Catalog 6008289) with assay buffer consisting of 50 mM Hepes ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095438(CHEMBL3589042)
Affinity DataIC50: 26nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50095350(CHEMBL3589034)
Affinity DataIC50: 27nMAssay Description:Inhibition of N-terminal GST tagged full-length human PRMT1 expressed in high five insect cells pre-incubated for 30 mins before addition of a [3H]SA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM502127(US11028083, Example 94b)
Affinity DataIC50: 27nMAssay Description:This enzymatic assay was performed in a 384 well, white, low volume plate (PerkinElmer, Catalog 6008289) with assay buffer consisting of 50 mM Hepes ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetProtein arginine N-methyltransferase 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM502129(US11028083, Example 95b)
Affinity DataIC50: 27nMAssay Description:This enzymatic assay was performed in a 384 well, white, low volume plate (PerkinElmer, Catalog 6008289) with assay buffer consisting of 50 mM Hepes ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

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