Compile Data Set for Download or QSAR
Report error Found 27 of affinity data for UniProtKB/TrEMBL: Q96PF2
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human TSSK2 using KKKVSRSGLYRSPSMPENLNRPR as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human TSSK2 using KKKVSRSGLYRSPSMPENLNRPR as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50329197(3-((R)-1-((2S,6R)-2,6-dimethylmorpholino)ethyl)-N-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50392791(CHEMBL2151321 | US8486966, 1)
Affinity DataIC50: 30.6nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50335188(CHEMBL1650551 | CHEMBL1650545 | N-[3-[(3,3-Difluor...)
Affinity DataIC50: 100nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50335188(CHEMBL1650551 | CHEMBL1650545 | N-[3-[(3,3-Difluor...)
Affinity DataIC50: 100nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50329198(CHEMBL1650533 | 2-{ethyl[(5-{[6-methyl-3-(1H-pyraz...)
Affinity DataIC50: 100nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50460773(CHEMBL4227082)
Affinity DataIC50: 500nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50460767(CHEMBL4228240)
Affinity DataIC50: 500nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50582077(CHEMBL5085753)
Affinity DataIC50: 944nMAssay Description:Inhibition of TSSK2 (unknown origin) by Z-lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50462709(CHEMBL4245507)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50433476(CHEMBL2381116)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50519662(CHEMBL4438748)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full-length human TSSK2 using KKKVSRSGLYRSP as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TSSK2 using [KKKVSRSGLYRSPSMPENLNRPR] as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/27/2017
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50499634(CHEMBL3741589)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50348621(CHEMBL1270795)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50433761(CHEMBL2381601)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50359359(CHEMBL1929238)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50362169(CHEMBL1938680)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50434485(CHEMBL2385543)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50045370(CHEMBL3314140)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50030881(CHEMBL3356117)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2016
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human His-tagged STK22B expressed in baculovirus expression system using serine/threonine-04 peptide as substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50224883(7-chloro-3-oxo-8-[(thiazol-5-ylmethyl)-amino]-11,1...)
Affinity DataKi: >1.53E+3nMAssay Description:Inhibition of TSSK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50463483(CHEMBL4245242)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTestis-specific serine/threonine-protein kinase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50463479(CHEMBL4249925)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of TSSK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed