Compile Data Set for Download or QSAR
Report error Found 15 of affinity data for UniProtKB/TrEMBL: Q93086
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118219(Bz-ATP | CHEMBL339386)
Affinity DataEC50:  4.00E+4nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 5 (P2X5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50598317(CHEMBL5208562)
Affinity DataIC50: 1.65E+3nMAssay Description:Antagonist activity against human P2X5R stably transfected in human 1321N1 cells incubated for 30 mins by Fura-2 AM staining based calcium influx ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50596631(CHEMBL1615626)
Affinity DataIC50: 7.01E+3nMAssay Description:Antagonist activity at human P2X5 receptor expressed in human 1321N1 cells assessed as reduction in intracellular Ca2+ influx incubated for 30 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50540409(CHEBI:34941 | CHEMBL69234)
Affinity DataIC50: 8.45E+3nMAssay Description:Antagonist activity against human P2X5R stably transfected in human 1321N1 cells incubated for 30 mins by Fura-2 AM staining based calcium influx ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50596630(CHEMBL5172961)
Affinity DataIC50: 9.04E+3nMAssay Description:Antagonist activity at human P2X5 receptor expressed in human 1321N1 cells assessed as reduction in intracellular Ca2+ influx incubated for 30 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50257829(Ro-51 | 2-(4-amino-5-(5-iodo-2-isopropyl-4-methoxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2X5 receptor up to 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50257636(5-(5-iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of P2X5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50415550(Ro-85 | CHEMBL599760)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2X5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50415563(CHEMBL605325)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at P2X5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50499490(CHEMBL3741992)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of P2X5R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50596625(CHEMBL5174645)
Affinity DataIC50: 1.23E+4nMAssay Description:Antagonist activity at human P2X5 receptor expressed in human 1321N1 cells assessed as reduction in intracellular Ca2+ influx incubated for 30 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataIC50: 1.58E+4nMAssay Description:Antagonist activity against human P2X5R stably transfected in human 1321N1 cells incubated for 30 mins by Fura-2 AM staining based calcium influx ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataIC50: 1.61E+4nMAssay Description:Antagonist activity at human P2X5 receptor expressed in human 1321N1 cells assessed as reduction in intracellular Ca2+ influx incubated for 30 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50596629(CHEMBL5200337)
Affinity DataIC50: 1.65E+4nMAssay Description:Antagonist activity at human P2X5 receptor expressed in human 1321N1 cells assessed as reduction in intracellular Ca2+ influx incubated for 30 mins b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetP2X purinoceptor 5(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50598315(CHEMBL5186938)
Affinity DataIC50: 2.76E+4nMAssay Description:Antagonist activity against human P2X5R stably transfected in human 1321N1 cells incubated for 30 mins by Fura-2 AM staining based calcium influx ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed