Compile Data Set for Download or QSAR
Report error Found 12 of affinity data for UniProtKB/TrEMBL: Q8NFI3
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50304533(2-((5R,6S,7R,8S)-8-acetamido-6,7-dihydroxy-5-methy...)
Affinity DataIC50: 1.83nMAssay Description:Inhibition of human placenta beta-N-acetylglucosaminidase by pNP-GlcNAc substrate hydrolysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50304532((1R*, 3S*, 5S*, 6S*, 7R*, 7a S*)-5-acetamidomethyl...)
Affinity DataIC50: 2.39nMAssay Description:Inhibition of human placenta beta-N-acetylglucosaminidase by pNP-GlcNAc substrate hydrolysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50373151(CHEMBL259756)
Affinity DataIC50: 420nMAssay Description:Inhibition of human endo-beta-N-acetylglucosaminidase expressed in Hek293 cells after 3 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50070209(CHEBI:8768 | Aciphex | LY-307640 | Rabeprazole)
Affinity DataIC50: 4.47E+3nMAssay Description:Inhibition of recombinant human C-MYC/DDK-tagged ENGase expressed in HEK293T cells using heat inactivated bovine ribonuclease B as substrate pretreat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2019
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50402289(TENATOPRAZOLE)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human C-MYC/DDK-tagged ENGase expressed in HEK293T cells using heat inactivated bovine ribonuclease B as substrate pretreat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2019
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50070208(CHEBI:6375 | A-65006 | AG-1749 | Lansoprazole | Pr...)
Affinity DataIC50: 2.44E+4nMAssay Description:Inhibition of recombinant human C-MYC/DDK-tagged ENGase expressed in HEK293T cells using heat inactivated bovine ribonuclease B as substrate pretreat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2019
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50247930(Dexilant | Dexilant solutab | Dexlansoprazole | Ka...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human C-MYC/DDK-tagged ENGase expressed in HEK293T cells using heat inactivated bovine ribonuclease B as substrate pretreat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2019
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50103597(CHEBI:77260 | Antra | H 168/68 | H-168/68 | Losec ...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human C-MYC/DDK-tagged ENGase expressed in HEK293T cells using heat inactivated bovine ribonuclease B as substrate pretreat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2019
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50235890((2S,3S)-3-Hydroxybaikiain | (2S,3S)-3-hydroxy-1,2,...)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibition of human placenta beta-N-acetylglucosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50235890((2S,3S)-3-Hydroxybaikiain | (2S,3S)-3-hydroxy-1,2,...)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibition of human Placental beta-N-acetylglucosaminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50304533(2-((5R,6S,7R,8S)-8-acetamido-6,7-dihydroxy-5-methy...)
Affinity DataKi:  0.925nMAssay Description:Competitive inhibition of human placenta beta-N-acetylglucosaminidase by pNP-GlcNAc substrate hydrolysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCytosolic endo-beta-N-acetylglucosaminidase(Human)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50304532((1R*, 3S*, 5S*, 6S*, 7R*, 7a S*)-5-acetamidomethyl...)
Affinity DataKi:  1.25nMAssay Description:Mixed type inhibition of human placenta beta-N-acetylglucosaminidase by pNP-GlcNAc substrate hydrolysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed