Compile Data Set for Download or QSAR
Report error Found 273 of affinity data for UniProtKB/TrEMBL: Q8MMZ8
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210476((2,5-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50: 0.0260nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50: 0.0400nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265424(2-{4-[3-(2-Aminopyrimidin-4-yl)-2-(4-fluorophenyl)...)
Affinity DataIC50: 0.0440nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50: 0.0440nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182369(4-(2-(4-fluorophenyl)-7-(1-methylpiperidin-4-yl)H-...)
Affinity DataIC50: 0.0440nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50168170(3-{4-[5-(4-Fluoro-phenyl)-4-pyridin-4-yl-1H-pyrrol...)
Affinity DataIC50: 0.0460nMAssay Description:In vitro inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182367(4-(2-(4-fluorophenyl)-7-(piperidin-4-yl)H-imidazo[...)
Affinity DataIC50: 0.0460nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182367(4-(2-(4-fluorophenyl)-7-(piperidin-4-yl)H-imidazo[...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50211814(4-(2-(4-fluorophenyl)-7-((isopropylamino)methyl)H-...)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210490((2-chlorobenzyl)-{4-[7-dimethylaminomethyl-2-(4-fl...)
Affinity DataIC50: 0.0560nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50211811(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210473((3,4-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210479((2,6-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210495(cyclopropylmethyl{4-[7-dimethylaminomethyl-2-(4-fl...)
Affinity DataIC50: 0.0640nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265425(2-{4-[3-(2-Aminopyrimidin-4-yl)-2-(4-fluorophenyl)...)
Affinity DataIC50: 0.0650nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265419(4-[7-(1-Dimethylaminobutyl)-2-(4-fluorophenyl)imid...)
Affinity DataIC50: 0.0650nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210517({4-[7-dimethylaminomethyl-2-(4-fluorophenyl)imidaz...)
Affinity DataIC50: 0.0660nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265397(4-[7-(1-Dimethylaminoethyl)-2-(4-fluorophenyl)imid...)
Affinity DataIC50: 0.0670nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265397(4-[7-(1-Dimethylaminoethyl)-2-(4-fluorophenyl)imid...)
Affinity DataIC50: 0.0670nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50211805(4-(7-(((3-(dimethylamino)propyl)(methyl)amino)meth...)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265430(4-[2-(4-Fluorophenyl)-7-(1-phenethylpiperidin-4-yl...)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50374578(CHEMBL401749)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210494({4-[7-dimethylaminomethyl-2-(4-fluorophenyl)imidaz...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210508(cyclopropyl{4-[7-dimethylaminomethyl-2-(4-fluoroph...)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50374594(CHEMBL444009)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182359(N-benzyl-4-(7-((dimethylamino)methyl)-2-(4-fluorop...)
Affinity DataIC50: 0.0810nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182359(N-benzyl-4-(7-((dimethylamino)methyl)-2-(4-fluorop...)
Affinity DataIC50: 0.0810nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210489({4-[7-dimethylaminomethyl-2-(4-fluorophenyl)imidaz...)
Affinity DataIC50: 0.0830nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210493({4-[7-dimethylaminomethyl-2-(4-fluorophenyl)imidaz...)
Affinity DataIC50: 0.0870nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210478({4-[7-dimethylaminomethyl-2-(4-fluorophenyl)imidaz...)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265427(4-[7-(1-Cyclopropylmethylpiperidin-4-yl)-2-(4-fluo...)
Affinity DataIC50: 0.0950nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50195444(2-(ethyl((2-(4-fluorophenyl)-3-(2-((S)-1-phenyleth...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50211820(4-(7-(((2-(azetidin-1-yl)ethyl)(methyl)amino)methy...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210500({4-[7-dimethylaminomethyl-2-(4-fluorophenyl)imidaz...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210511(4-[2-(2,4-difluorophenyl)-7-dimethylaminomethylimi...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50248496(2-(4-(2-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-indol...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of Eimeria tenella parasite-specific cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210514(cyclopentyl{4-[7-dimethylaminomethyl-2-(4-fluoroph...)
Affinity DataIC50: 0.102nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182362(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)imi...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50195435(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethyl)py...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Eimeria tenella PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50211802(2-(((2-(4-fluorophenyl)-3-(2-((S)-1-phenylethylami...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50211812(4-(2-(4-fluorophenyl)-7-((isopropyl(methyl)amino)m...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Et-PKGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210486((3,5-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265404(4-(7-(1-ethylpiperidin-4-yl)-2-(4-fluorophenyl)imi...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265429(4-[7-(1-Benzylpiperidin-4-yl)-2-(4-fluorophenyl)-i...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265402(4-[7-[1-(3,3-Dimethylbutyl)piperidin-4-yl)-2-(4-fl...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265421(4-[7-(1-Dimethylamino-1-methyl-ethyl)-2-(4-fluorop...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50182362(4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)imi...)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210488((2,3-difluorobenzyl)-{4-[7-dimethylaminomethyl-2-(...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50210505(cyclohexyl-{4-[7-dimethylaminomethyl-2-(4-fluoroph...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinase by Ten_K assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcGMP-dependent protein kinase(Coccidian parasite)
Scynexis

Curated by ChEMBL
LigandPNGBDBM50265403(4-{2-(4-Fluorophenyl)-7-[1-(2-methylpentyl)piperid...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of Eimeria tenella cGMP-dependent protein kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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