Compile Data Set for Download or QSAR
Report error Found 18 of affinity data for UniProtKB/TrEMBL: Q8CFK4
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50013712(Pyridin-2-ylamine | 2-aminopyridine | CHEMBL21619 ...)
Affinity DataKd: >4.00E+6nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154591(6-Bromo-quinolin-2-ylamine | CHEMBL189197)
Affinity DataEC50:  5.80E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154582(6-[1,3]Dioxan-2-yl-quinolin-2-ylamine | CHEMBL4266...)
Affinity DataKd:  5.20E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154587(6-[1,3]Dioxolan-2-yl-quinolin-2-ylamine | CHEMBL36...)
Affinity DataEC50:  3.40E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154589(6-Chloro-quinolin-2-ylamine | CHEMBL189514)
Affinity DataEC50:  7.60E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154590(6-Methoxy-quinolin-2-ylamine | CHEMBL188730)
Affinity DataEC50:  6.30E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154588(5,6,7,8-Tetrahydro-quinolin-2-ylamine | CHEMBL1888...)
Affinity DataEC50:  2.15E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50084506(Methyl-quinolin-2-yl-amine | CHEMBL319543)
Affinity DataKd:  3.80E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154587(6-[1,3]Dioxolan-2-yl-quinolin-2-ylamine | CHEMBL36...)
Affinity DataKd:  4.00E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154582(6-[1,3]Dioxan-2-yl-quinolin-2-ylamine | CHEMBL4266...)
Affinity DataEC50:  2.60E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM14320(CHEMBL62083 | 1-amino-isoquinoline | fragment 1 (J...)
Affinity DataKd:  6.50E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM14322(CHEMBL61236 | 2-aminoquinoline | fragment 2 (J. me...)
Affinity DataEC50:  1.60E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154583(6-Methyl-quinolin-2-ylamine | CHEMBL361660)
Affinity DataEC50:  7.50E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154586(6-(5,5-Dimethyl-[1,3]dioxan-2-yl)-quinolin-2-ylami...)
Affinity DataKd:  2.20E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154585(Quinazolin-2-ylamine | CHEMBL187951)
Affinity DataKd:  8.00E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154584(6-Fluoro-quinolin-2-ylamine | CHEMBL185917)
Affinity DataEC50:  1.50E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM50154583(6-Methyl-quinolin-2-ylamine | CHEMBL361660)
Affinity DataKd:  6.10E+4nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase(Mouse)
The University of Adelaide

Curated by ChEMBL
LigandPNGBDBM14322(CHEMBL61236 | 2-aminoquinoline | fragment 2 (J. me...)
Affinity DataKd:  1.25E+5nMAssay Description:Displacement of PRP-1 peptide from mouse Tec kinase SH3 domain by fluorescence polarizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed