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Report error Found 5 for UniProtKB: Q8BLD9
TargetD(1B) dopamine receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM435739(US10611751, Example 1 | 2-(2,6-dichlorophenyl)-1-(...)
Affinity DataEC50:  480nMAssay Description:Positive allosteric modulation of mouse D5 receptor expressed in HEK293 cells assessed as increase in cyclic AMP production measured after 60 mins in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetD(1B) dopamine receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM435739(US10611751, Example 1 | 2-(2,6-dichlorophenyl)-1-(...)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at mouse D5 receptor expressed in HEK293 cells assessed as increase in cyclic AMP production measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Mouse)
Johns Hopkins Medical Institutions

Curated by ChEMBL
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataIC50: 3.50E+4nMAssay Description:Ability (10 ug/kg) to inhibit binding of [125I]iododexetimide to Dopamine receptor of miceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2019
Entry Details Article
PubMed
TargetD(1B) dopamine receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM186937(US9079895, 25s)
Affinity DataKi:  8.53E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
Go to US Patent

TargetD(1B) dopamine receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM186930(US9079895, 21s | US9079895, 20s)
Affinity DataKi: >1.00E+4nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
Go to US Patent