Compile Data Set for Download or QSAR
Report error Found 3 of affinity data for UniProtKB/TrEMBL: Q6R6I6
TargetRelaxin receptor 1(Rat)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563215(CHEMBL4781560)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Rat)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563220(CHEMBL4793799)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Rat)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563230(CHEMBL4754949)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed