Compile Data Set for Download or QSAR
Report error Found 353 of affinity data for UniProtKB/TrEMBL: Q6DWJ6
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131895(CHEMBL3633896)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131896(CHEMBL3633895)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131897(CHEMBL3633894)
Affinity DataEC50:  670nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131899(CHEMBL3633893)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131900(CHEMBL3633892)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131901(CHEMBL3633891)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131902(CHEMBL3633890)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131903(CHEMBL3633889)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131904(CHEMBL3633888)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131905(CHEMBL3633887)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131906(CHEMBL3633886)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131931(CHEMBL3633885)
Affinity DataEC50:  193nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131946(CHEMBL3633884)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131993(CHEMBL3633883)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131994(CHEMBL3633882)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50131999(CHEMBL3633881)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132000(CHEMBL3633880)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132131(CHEMBL3633879)
Affinity DataEC50:  59nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132137(CHEMBL3633878)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132141(CHEMBL3633721)
Affinity DataEC50:  118nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50132143(CHEMBL3633720)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human GPR139 receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263505(n-(4-chlorophenethyl)-2-(4-oxobenzo[d][1,2,3]triaz...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566727(CHEMBL1310918)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566728(CHEMBL4866435)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263506(n-(3-chlorophenethyl)-2-(4-oxobenzo[d][1,2,3]triaz...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566729(CHEMBL1380104)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263507(n-(4-methylphenethyl)-2-(4-oxobenzo[d][1,2,3]triaz...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566730(CHEMBL4869485)
Affinity DataEC50:  85nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263508((r)-2-(4-oxobenzo[d][1,2,3]triazin-3(4h)-yl)-n-(2-...)
Affinity DataEC50:  288nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566731(CHEMBL4856162)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263510((s)-n-(1-(4-methoxyphenyl)propan-2-yl)-2-(4-oxoben...)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566732(CHEMBL4852809)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566733(CHEMBL4878791)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566734(CHEMBL1546963)
Affinity DataEC50:  293nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566735(CHEMBL4860510)
Affinity DataEC50:  79nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263391((s)-n-(1-(4-chlorophenyl)ethyl)-2-(4-oxobenzo[d][1...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263433((s)-2-(4-oxobenzo[d][1,2,3]triazin-3(4h)-yl)-n-(1-...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566736(CHEMBL4874254)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263370((s)-2-(4-oxobenzo[d][1,2,3]triazin-3(4h)-yl)-n-(1-...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566737(CHEMBL4788631)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566738(CHEMBL4861019)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263385((s)-n-(1-(4-methoxyphenyl)ethyl)-2-(4-oxobenzo[d][...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263435((s)-n-(1-(4-ethoxyphenyl)ethyl)-2-(4-oxobenzo[d][1...)
Affinity DataEC50:  67nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566739(CHEMBL4792727)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566740(CHEMBL4776509)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566741(CHEMBL4856133)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50566742(CHEMBL4852265)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263420((s)-n-(1-(2,4-dimethylphenyl)ethyl)-2-(4-oxobenzo[...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263485((s)-n-(1-(2-fluoro-4-methylphenyl)ethyl)-2-(4-oxob...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 139(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM263483((s)-n-(1-(2-methoxy-4-methylphenyl)ethyl)-2-(4-oxo...)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
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