Compile Data Set for Download or QSAR
Report error Found 11 of affinity data for UniProtKB/TrEMBL: Q6B4J2
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50166637(2'-Biphenyl-4-yl-4-hydroxy-3',4'-dihydro-2'H-[3,4'...)
Affinity DataIC50: 40nMAssay Description:Inhibitory concentration against beef liver Vitamin K epoxide reductase (vitamin K 2,3-epoxide reductase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50166638(13-(4-phenylphenyl)-4,12,14-trioxapentacyclo[11.7....)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against beef liver Vitamin K epoxide reductase (vitamin K 2,3-epoxide reductase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50015554(CHEMBL51057 | 7a-Hydroxymethyl-1a-(3,7,11,15-tetra...)
Affinity DataKi:  8.00E+3nMAssay Description:Apparent kinetic constant for Vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50018515(CHEMBL67386 | 2-Fluoromethyl-2-hydroxy-3-methyl-3-...)
Affinity DataKi:  1.60E+4nMAssay Description:Binding affinity for vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50015552(CHEMBL51260 | 7a-Fluoromethyl-1a-(3,7,11,15-tetram...)
Affinity DataKi:  1.70E+4nMAssay Description:Apparent kinetic constant for Vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50015556(CHEMBL51080 | 2,7-Dioxo-1a-(3,7,11,15-tetramethyl-...)
Affinity DataKi:  2.60E+4nMAssay Description:Apparent kinetic constant for Vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50015559(CHEMBL297521 | 1a-(1-Hydroxy-3,7,11,15-tetramethyl...)
Affinity DataKi:  4.30E+4nMAssay Description:Apparent kinetic constant for Vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50015555(CHEMBL52683 | 7a-Difluoromethyl-1a-(3,7,11,15-tetr...)
Affinity DataKi:  6.30E+4nMAssay Description:Apparent kinetic constant for Vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50015557(CHEMBL51180 | 1a-(1-Hydroxy-3,7,11,15-tetramethyl-...)
Affinity DataKi:  6.30E+4nMAssay Description:Apparent kinetic constant for Vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50015553(CHEMBL53971 | 7a-Chloromethyl-1a-(3,7,11,15-tetram...)
Affinity DataKi:  7.40E+4nMAssay Description:Apparent kinetic constant for Vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVitamin K epoxide reductase complex subunit 1(Bovine)
Tunghai University

Curated by ChEMBL
LigandPNGBDBM50015558(CHEMBL50340 | 1a-(1-Fluoro-3,7,11,15-tetramethyl-h...)
Affinity DataKi:  1.00E+5nMAssay Description:Apparent kinetic constant for Vitamin K epoxide reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed