Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataEC50: 107nMAssay Description:Agonist activity at mouse 5-HT1A expressed in HEK293 cells after 2 to 5 minsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Compound was evaluated for the affinity at 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor was determined using [3H]-8-OH-DPAT radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 238nMAssay Description:Compound was tested for the binding affinity against 5-hydroxytryptamine 1A receptor by using [3H]DPAT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Compound was evaluated for the affinity at 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of 5-OH-DPAT binding to 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against serotonin 5-hydroxytryptamine 1A receptor from mice.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 9.10E+3nMAssay Description:Ability to displace [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 3.58E+5nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Compound was evaluated for the binding affinity against [3H]8-OH-DPAT-labeled 5-hydroxytryptamine 1A receptor sites in cloned CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Compound was evaluated for the binding affinity against [3H]8-OH-DPAT-labeled 5-hydroxytryptamine 1A receptor sites in cloned CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.600nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Mouse)
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Julius Maximilian University of W£Rzburg
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Ability to displace [125I]iodosulpiride from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
