Compile Data Set for Download or QSAR
Report error Found 81 of affinity data for UniProtKB/TrEMBL: Q64077
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217519(CHEMBL354709)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50403793(CHEMBL2115415)
Affinity DataIC50: 3.10nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217520(CHEMBL354645)
Affinity DataIC50: 3.20nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217517(CHEMBL353158)
Affinity DataIC50: 4.70nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217506(CHEMBL170936)
Affinity DataIC50: 5.5nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217504(CHEMBL353284)
Affinity DataIC50: 6.20nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217513(CHEMBL171658)
Affinity DataIC50: 6.80nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50090485(spiro[(2-hydroxy)indane-1,40-piperidine] analogue ...)
Affinity DataIC50: 6.80nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217528(CHEMBL353596)
Affinity DataIC50: 6.90nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217509(CHEMBL354731)
Affinity DataIC50: 7.30nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217505(CHEMBL414377)
Affinity DataIC50: 7.5nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217527(CHEMBL172227)
Affinity DataIC50: 9.30nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217514(CHEMBL369246)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217529(CHEMBL171719)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217512(CHEMBL169132)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217510(CHEMBL355387)
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217507(CHEMBL171704)
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50090487(spiro[(2-hydroxy)indane-1,40-piperidine] analogue ...)
Affinity DataIC50: 45nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217523(CHEMBL353168)
Affinity DataIC50: 52nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50403790(CHEMBL2114963)
Affinity DataIC50: 59nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217522(CHEMBL353394)
Affinity DataIC50: 64nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217518(CHEMBL353480)
Affinity DataIC50: 74nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217526(CHEMBL366972)
Affinity DataIC50: 89nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217508(CHEMBL367509)
Affinity DataIC50: 91nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217521(CHEMBL355310)
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217511(CHEMBL172342)
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217525(CHEMBL171414)
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217515(CHEMBL352350)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217530(CHEMBL170084)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217531(CHEMBL170083)
Affinity DataIC50: 440nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50217516(CHEMBL354288)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against Neurokinin 2 (NK2) receptor from guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2018
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50403792(CHEMBL2115416)
Affinity DataIC50: 1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50403791(CHEMBL2114965)
Affinity DataIC50: 1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50090484(spiro[(2-hydroxy)indane-1,40-piperidine] analogue ...)
Affinity DataIC50: 1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50090482(spiro[(2-hydroxy)indane-1,40-piperidine] analogue ...)
Affinity DataIC50: 1.00E+3nMAssay Description:The compound was evaluated in vitro for its ability to displace [3H]SP from Tachykinin receptor 2 of male guinea pig lung membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116083(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116074(N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']bipiperidinyl-...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116091(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116076(N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']bipiperidinyl-...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116082(3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2...)
Affinity DataKi:  0.300nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116080(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116078(CHEMBL66332 | SCH 206272 | 3,5-Dichloro-N-[3-(3,4-...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116088(3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116090(1-(2-{1'-[5-[(3,5-Dichloro-benzoyl)-ethyl-amino]-3...)
Affinity DataKi:  0.700nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116075(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116075(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116087(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116085(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.900nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116089(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  1nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSubstance-K receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50116077(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  1nMAssay Description:In vitro binding to Tachykinin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
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