Compile Data Set for Download or QSAR
Report error Found 13 of affinity data for UniProtKB/TrEMBL: Q63449
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataEC50:  16nMAssay Description:Binding affinity to progesterone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50107347(5-Allyl-10-methoxy-2,2,4-trimethyl-2,5-dihydro-1H-...)
Affinity DataEC50:  126nMAssay Description:Binding affinity to progesterone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50366382(CHEMBL57078)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]R5020 binding to cytosolic progesterone receptor (PRc) of rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of [3H]R5020 binding to cytosolic progesterone receptor (PRc) of rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50366381(CHEMBL301446)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of [3H]R5020 binding to cytosolic progesterone receptor (PRc) of rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50126158(3-fluoro-5-(2'-thioxo-1',2'-dihydrospiro[cyclohexa...)
Affinity DataIC50: 7.43nMAssay Description:Inhibitory progestational activity on oral administration in uterine C3 modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50366380(CHEMBL56509)
Affinity DataIC50: 9nMAssay Description:Inhibition of [3H]R5020 binding to cytosolic progesterone receptor (PRc) of rat uterusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50067678(17-Acetoxy-6alpha-methylprogesterone | 17alpha-Hyd...)
Affinity DataIC50: 67.3nMAssay Description:Inhibitory progestational activity on oral administration in uterine C3 modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50404222(CHEMBL417475)
Affinity DataIC50: 92.5nMAssay Description:Inhibitory progestational activity on oral administration in uterine C3 modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50375837(CHEMBL270976)
Affinity DataIC50: 942nMAssay Description:Inhibitory progestational activity on oral administration in uterine C3 modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM50404229(CHEMBL24089)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibitory progestational activity on oral administration in uterine C3 modelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM18656((2R,5S)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-...)
Affinity DataKi:  3.30E+3nMAssay Description:Activities of the test compounds to inhibit androgen receptor mediated transcription induced by DHT were evaluated using stable transfected AR/CHO#3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2007
Entry Details Article
PubMed
TargetProgesterone receptor(Rat)
Forschungszentrum Dresden-Rossendorf

Curated by ChEMBL
LigandPNGBDBM18525(N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluoro...)
Affinity DataKi:  7.20E+3nMAssay Description:Activities of the test compounds to inhibit androgen receptor mediated transcription induced by DHT were evaluated using stable transfected AR/CHO#3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2007
Entry Details Article
PubMed