Compile Data Set for Download or QSAR
Report error Found 384 of affinity data for UniProtKB/TrEMBL: Q63380
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50176062(3-(5H-dibenzo[a,d][7]annulen-5-yl)-N-methylpropan-...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM35226(Vestra | Reboxetine | (S,S)-reboxetine)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50275774(N,N-Diallyl (1R,2R)-2-(Aminomethyl)-1-(2-thienyl)c...)
Affinity DataIC50: 4.60nMAssay Description:Displacement of Levo[ring-2,5,6-3H]norepinephrine from rat synaptosomal NET expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50239791((1S,2R)-N-allyl-2-(aminomethyl)-N-ethyl-1-(thiophe...)
Affinity DataIC50: 6.40nMAssay Description:Displacement of Levo[ring-2,5,6-3H]norepinephrine from rat synaptosomal NET expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50009717(CHEMBL436281)
Affinity DataIC50: 10nMAssay Description:Inhibition of NET-mediated norepinephrine uptake in rat brain synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50275831(2-[(1R,2R)-2-(Aminomethyl)-1-(2-thienyl)cyclopropa...)
Affinity DataIC50: 15nMAssay Description:Displacement of Levo[ring-2,5,6-3H]norepinephrine from rat synaptosomal NET expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50275771(1S,2R-milnacipran | CHEMBL471001)
Affinity DataIC50: 16nMAssay Description:Displacement of Levo[ring-2,5,6-3H]norepinephrine from rat synaptosomal NET expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50275773(N-Ethyl-N-(2-fluoroallyl) (1R,2R)-2-(Aminomethyl)-...)
Affinity DataIC50: 21nMAssay Description:Displacement of Levo[ring-2,5,6-3H]norepinephrine from rat synaptosomal NET expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM82217([4-(3,4-Dichloro-phenyl)-1,2,3,4-tetrahydro-naphth...)
Affinity DataIC50: 22nMAssay Description:Inhibition of [3H]norepinephrine reuptake at NET in rat brain synaptosome by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243939((cis)-1-(3,4-dichlorophenyl)-6-methyl-3-aza-bicycl...)
Affinity DataIC50: 29nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50032379((1S,2R)-2-Aminomethyl-1-phenyl-cyclopropanecarboxy...)
Affinity DataIC50: 30nMAssay Description:Displacement of Levo[ring-2,5,6-3H]norepinephrine from rat synaptosomal NET expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243940((cis)-1-(3,4-dichlorophenyl)-6-phenyl-3-aza-bicycl...)
Affinity DataIC50: 34nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243942(1-(naphthalen-2-yl)-3-aza-bicyclo[3.1.0]hexane | C...)
Affinity DataIC50: 36nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243986(1-(benzofuran-2-yl)-3-aza-bicyclo[3.1.0]hexane | C...)
Affinity DataIC50: 48nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243937((1R,5S)-1-(3,4-dichlorophenyl)-3-aza-bicyclo[3.1.0...)
Affinity DataIC50: 51nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243987(1-(benzo[b]thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexa...)
Affinity DataIC50: 53nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50244081((1S,5S)-1-(5-fluorobenzo[b]thiophen-2-yl)-3-aza-bi...)
Affinity DataIC50: 67nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50244040((1S,5S)-1-(5-chlorothiophen-2-yl)-3-aza-bicyclo[3....)
Affinity DataIC50: 77nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243895(1-(3,4-dichlorophenyl)-3-aza-bicyclo[3.1.0]hexane ...)
Affinity DataIC50: 88nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243991((1S,5S)-1-(thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexa...)
Affinity DataIC50: 92nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50032379((1S,2R)-2-Aminomethyl-1-phenyl-cyclopropanecarboxy...)
Affinity DataIC50: 100nMAssay Description:Inhibition of radiolabeled noradrenaline uptake from rat brain NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243894((cis)-1,6-diphenyl-3-aza-bicyclo[3.1.0]hexane | CH...)
Affinity DataIC50: 120nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243989(1-(thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexane | CHE...)
Affinity DataIC50: 130nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50244082(1-(5-chlorothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexa...)
Affinity DataIC50: 130nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243889((cis)-2-methyl-1-(thiophen-2-yl)-3-aza-bicyclo[3.1...)
Affinity DataIC50: 150nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243990((1R,5R)-1-(thiophen-2-yl)-3-aza-bicyclo[3.1.0]hexa...)
Affinity DataIC50: 150nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50010858(CHEMBL101899 | 1-[1-(3-Chloro-phenyl)-2-dimethylam...)
Affinity DataIC50: 160nMAssay Description:Inhibition of norepinephrine uptake at rat brain norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50275829(N-Ethyl-N-propargyl (1R,2R)-2-(Aminomethyl)-1-(2-t...)
Affinity DataIC50: 160nMAssay Description:Displacement of Levo[ring-2,5,6-3H]norepinephrine from rat synaptosomal NET expressed in HEK293 cells by microplate scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50309172((1R,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 185nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50244041(1-(5-bromothiophen-2-yl)-3-aza-bicyclo[3.1.0]hexan...)
Affinity DataIC50: 190nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50005246(beta-aminopropylbenzene | AMPHETAMINE SULFATE | de...)
Affinity DataIC50: 200nMAssay Description:Inhibition of [3H]norepinephrine uptake at NET expressed in rat hypothalamic homogenate containing synaptosomes after 5 mins by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243988(1-(benzo[b]thiophen-3-yl)-3-aza-bicyclo[3.1.0]hexa...)
Affinity DataIC50: 220nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50010874(1-[1-(4-Chloro-phenyl)-2-dimethylamino-ethyl]-cycl...)
Affinity DataIC50: 300nMAssay Description:Inhibition of norepinephrine uptake at rat brain norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50244046((1S,5R)-1-(thiophen-3-yl)-3-aza-bicyclo[3.1.0]hexa...)
Affinity DataIC50: 300nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243992((trans)-4-methyl-1-(thiophen-2-yl)-3-aza-bicyclo[3...)
Affinity DataIC50: 320nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50244045((1R,5R)-1-(5-bromothiophen-2-yl)-3-aza-bicyclo[3.1...)
Affinity DataIC50: 340nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243891(1-phenyl-3-aza-bicyclo[3.1.0]hexane | CHEMBL503383)
Affinity DataIC50: 350nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50010884(CHEMBL99653 | 1-[2-Dimethylamino-1-(3-trifluoromet...)
Affinity DataIC50: 360nMAssay Description:Inhibition of norepinephrine uptake at rat brain norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243943(1-Biphenyl-4-yl-3-aza-bicyclo[3.1.0]hexane | CHEMB...)
Affinity DataIC50: 360nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50309173(rac-erythro-2-(4-benzylpiperazin-1-yl)-1-(5-chloro...)
Affinity DataIC50: 425nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243896((1S,5R)-1-(3,4-dichlorophenyl)-3-aza-bicyclo[3.1.0...)
Affinity DataIC50: 430nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50244049((1S,5S)-1-(5-fluorothiophen-2-yl)-3-aza-bicyclo[3....)
Affinity DataIC50: 470nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243938((trans)-1-(3,4-dichlorophenyl)-6-methyl-3-aza-bicy...)
Affinity DataIC50: 500nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243993((cis)-4-methyl-1-(thiophen-2-yl)-3-aza-bicyclo[3.1...)
Affinity DataIC50: 560nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50243995((1R,5R)-1-(5-chlorothiophen-2-yl)-3-aza-bicyclo[3....)
Affinity DataIC50: 590nMAssay Description:Inhibition of norepinephrine uptake at NET in rat brain synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50010879(1-(2-(dimethylamino)-1-(3-methoxyphenyl)ethyl)cycl...)
Affinity DataIC50: 620nMAssay Description:Inhibition of norepinephrine uptake at rat brain norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM82071(NSC_62923 | WY-45030 | VENLAFAXINE | CAS_93413-69-...)
Affinity DataIC50: 640nMAssay Description:Inhibition of norepinephrine uptake at rat brain norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50010860(1-(1-(2-chlorophenyl)-2-(dimethylamino)ethyl)cyclo...)
Affinity DataIC50: 640nMAssay Description:Inhibition of norepinephrine uptake at rat brain norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50309175((1R,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50386200(CHEMBL2043240)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat NET-mediated norepinephrine reuptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
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