Compile Data Set for Download or QSAR
Report error Found 95 for UniProtKB: Q62986
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228276(CHEMBL1627365)
Affinity DataEC50:  2.98E+3nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50227469(CHEMBL285536)
Affinity DataEC50:  2.90nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50227470(CHEMBL34648)
Affinity DataEC50:  4.5nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50227469(CHEMBL285536)
Affinity DataEC50:  170nMAssay Description:In vitro displacement of 3 nM [3H]4-hydroxytamoxifen from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50227468(CHEMBL33879)
Affinity DataEC50:  10nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataEC50:  1.83E+3nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228277(CHEMBL1627386)
Affinity DataEC50:  7.03E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50175410(4-(2-(1-methyl-1H-pyrrol-2-yl)-1H-benzo[d]imidazol...)
Affinity DataEC50:  40.8nMAssay Description:Effect on ERbeta in rat ovary granulosa cell line transfected with ER responsive luciferase reporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50175419(4-(2-phenyl-1H-indol-3-yl)phenol | CHEMBL371012)
Affinity DataEC50:  1.09nMAssay Description:Effect on ERbeta in rat ovary granulosa cell line transfected with ER responsive luciferase reporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataEC50:  0.140nMAssay Description:Effect on ERbeta in rat ovary granulosa cell line transfected with ER responsive luciferase reporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50175415(4-(5-phenyl-2-(trifluoromethyl)-1H-imidazol-4-yl)p...)
Affinity DataEC50:  6.70nMAssay Description:Effect on ERbeta in rat ovary granulosa cell line transfected with ER responsive luciferase reporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataEC50:  5.70nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228273(CHEMBL1627375)
Affinity DataEC50:  1.92E+4nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228275(CHEMBL1627370)
Affinity DataEC50:  5.12E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228274(CHEMBL1627389)
Affinity DataEC50:  1.86E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228273(CHEMBL1627375)
Affinity DataEC50:  5.76E+4nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50187243(ethinyloestradiol | 17alpha-ethynylestra-1,3,5(10)...)
Affinity DataEC50:  1.68E+3nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228275(CHEMBL1627370)
Affinity DataEC50:  1.66E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50187243(ethinyloestradiol | 17alpha-ethynylestra-1,3,5(10)...)
Affinity DataEC50: >3.37E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50228277(CHEMBL1627386)
Affinity DataEC50:  2.81E+4nMAssay Description:Displacement of [3H]-estradiol from estrogen receptor in mature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataEC50:  917nMAssay Description:Displacement of [3H]estradiol from estrogen receptor in immature ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/9/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50225311(CHEMBL15128)
Affinity DataKd:  220nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50225310(CHEMBL1794824)
Affinity DataKd:  160nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50023749(4-[1-(4-hydroxyphenyl)-2-phenylvinyl]phenol | 4-(1...)
Affinity DataEC50:  3.20nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM8903(CHEMBL103 | (1S,2R,10S,11S,14S,15S)-14-acetyl-2,15...)
Affinity DataKd:  3.90nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50225312(CHEMBL14506)
Affinity DataKd:  730nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM20608([3H]4-OHT | cid_449459 | CHEMBL489 | AFIMOXIFENE |...)
Affinity DataEC50:  6nMAssay Description:In vitro displacement of 3 nM [3H]4-hydroxytamoxifen from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50148732(17alpha-ethinyl-19-nortestosterone | 17alpha-ethin...)
Affinity DataKd:  0.630nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50227471(CHEMBL287352)
Affinity DataEC50:  9.5nMAssay Description:In vitro displacement of 3 nM [3H]4-hydroxytamoxifen from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50225313(CHEMBL273571)
Affinity DataKd:  5.10E+3nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50227471(CHEMBL287352)
Affinity DataEC50:  3.30nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50225314(CHEMBL1627822)
Affinity DataKd:  0.620nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 0.354nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50123205(2-(4-hydroxyphenyl)-1,2'-spirobi[1H-indene]-5-ol |...)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity foor Rat Estrogen receptor-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50154088(7-bromo-2-(4-hydroxyphenyl)benzo[d]oxazol-5-ol | 7...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50123208(2-(4-hydroxyphenyl)-3-methyl-1,2'-spirobi[1H-inden...)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity foor Rat Estrogen receptor-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]- Estradiol from Estrogen receptor of rat uterine cytosolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM19441(Evista | CHEMBL81 | Keoxifene | Raloxifene, 6 | RA...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50214281(MESO-HEXESTROL | Hexestrol)
Affinity DataIC50: 2nMAssay Description:Binding affinity for rat estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2018
Entry Details

TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50154084(7-bromo-2-(3-fluoro-4-hydroxyphenyl)benzo[d]oxazol...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 2nMAssay Description:Binding affinity for Estrogen receptor beta(ER beta) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50154057(2-(4-hydroxyphenyl)benzo[d]oxazol-5-ol | 2-(4-Hydr...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50123209(5'-(2-hexahydro-1-pyridinylethoxy)-2-(4-hydroxyphe...)
Affinity DataIC50: 2.70nMAssay Description:Binding affinity foor Rat Estrogen receptor-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50154055(2-(3-FLUORO-4-HYDROXYPHENYL)-7-VINYL-1,3-BENZOXAZO...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM19441(Evista | CHEMBL81 | Keoxifene | Raloxifene, 6 | RA...)
Affinity DataIC50: 3.40nMAssay Description:Binding affinity foor Rat Estrogen receptor-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50154045(5-hydroxy-2-(4-hydroxyphenyl)benzo[d]oxazole-7-car...)
Affinity DataIC50: 4nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50054811({4-[(Z)-1-(4-Hydroxy-phenyl)-2-phenyl-but-1-enyl]-...)
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]- Estradiol from Estrogen receptor of rat uterine cytosolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM50471710(CHEMBL317748)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Sri International

Curated by ChEMBL
LigandPNGBDBM20606((5R,6S)-6-phenyl-5-[4-(2-pyrrolidin-1-ylethoxy)phe...)
Affinity DataIC50: 11nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 95 total ) | Next | Last >>
Jump to: