Compile Data Set for Download or QSAR
Report error Found 444 for UniProtKB: Q62758
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000480nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(GR-125487 | 5-Fluoro-2-methoxy-1H-indole-3-carboxy...)
Affinity DataKi:  0.000910nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(SB-207266 | N-(1-Butylpiperidine-4-ylmethyl)-1,2-(...)
Affinity DataKi:  0.00560nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85020(GR-125487 | 5-Fluoro-2-methoxy-1H-indole-3-carboxy...)
Affinity DataKi:  0.00890nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105635(6-Chloro-1H-benzoimidazole-4-carboxylic acid [1-(2...)
Affinity DataKi:  0.110nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]GR-113808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105635(6-Chloro-1H-benzoimidazole-4-carboxylic acid [1-(2...)
Affinity DataKi:  0.110nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50288595(4-Amino-5-chloro-2,3-dihydro-benzofuran-7-carboxyl...)
Affinity DataKi:  0.130nMAssay Description:Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatum by [3H]GR-113808 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatal membranes by [3H]GR-113808 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29525(GR 113808 | [3H] GR 113808 | CHEMBL518682 | 3H-GR1...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50007872(BIMU 1 | CHEMBL62023 | CHEMBL544755 | 3-Ethyl-2-ox...)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50058173(CHEMBL50660 | ML10375 | 4-Amino-5-chloro-2-methoxy...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatal membranes by [3H]GR-113808 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105650(6-Chloro-1H-benzoimidazole-4-carboxylic acid (1-is...)
Affinity DataKi:  0.290nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105650(6-Chloro-1H-benzoimidazole-4-carboxylic acid (1-is...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]GR-113808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398598(CHEMBL2152922)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]GR113808 from 5HT4 receptor in rat striatal membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105649(6-Chloro-1H-benzoimidazole-4-carboxylic acid (1-bu...)
Affinity DataKi:  0.320nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105649(6-Chloro-1H-benzoimidazole-4-carboxylic acid (1-bu...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]GR-113808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  0.390nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85026(SB-207266 | N-(1-Butylpiperidine-4-ylmethyl)-1,2-(...)
Affinity DataKi:  0.470nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/1/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105640(6-Chloro-1H-benzoimidazole-4-carboxylic acid (1-pe...)
Affinity DataKi:  0.540nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]GR-113808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105640(6-Chloro-1H-benzoimidazole-4-carboxylic acid (1-pe...)
Affinity DataKi:  0.540nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398598(CHEMBL2152922)
Affinity DataEC50:  0.590nMAssay Description:Agonist activity at rat 5HT4S receptor expressed in HEK293 cells assessed as increase in cAMP production after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398598(CHEMBL2152922)
Affinity DataEC50:  0.620nMAssay Description:Agonist activity at rat 5HT4E receptor expressed in HEK293 cells assessed as increase in cAMP production after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105653(6-Bromo-1H-benzoimidazole-4-carboxylic acid (1-but...)
Affinity DataKi:  0.640nMAssay Description:Binding affinity to 5-hydroxytryptamine 4 receptor using [3H]GR-113808 as radioligand in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50105653(6-Bromo-1H-benzoimidazole-4-carboxylic acid (1-but...)
Affinity DataKi:  0.640nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 4 receptor in rat striatum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398598(CHEMBL2152922)
Affinity DataEC50:  0.650nMAssay Description:Agonist activity at rat 5HT4L receptor expressed in HEK293 cells assessed as increase in cAMP production after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398590(CHEMBL2179583)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at rat 5HT4S receptor expressed in HEK293 cells assessed as increase in cAMP production after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056418(4-Amino-5-chloro-2-methoxy-benzoic acid 2-azepan-1...)
Affinity DataKi:  0.920nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056406(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-methy...)
Affinity DataKi:  0.930nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50288597(4-Amino-5-chloro-2,3-dihydro-benzofuran-7-carboxyl...)
Affinity DataKi:  0.940nMAssay Description:Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatum by [3H]GR-113808 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398590(CHEMBL2179583)
Affinity DataEC50:  0.960nMAssay Description:Agonist activity at rat 5HT4L receptor expressed in HEK293 cells assessed as increase in cAMP production after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056403(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(3-hydro...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50058170((2-Ethoxy-phenyl)-carbamic acid 2-((3R,5S)-3,5-dim...)
Affinity DataKi:  1.05nMAssay Description:Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatal membranes by [3H]GR-113808 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29526(CHEMBL286136 | 2-Piperidinoethyl 4-amino-5-chloro-...)
Affinity DataKi:  1.07nMAssay Description:Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatal membranes by [3H]GR-113808 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29526(CHEMBL286136 | 2-Piperidinoethyl 4-amino-5-chloro-...)
Affinity DataKi:  1.07nMAssay Description:Binding affinity against 5-hydroxytryptamine 4 receptor using [3H]GR-113808 as radioligand in rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM29526(CHEMBL286136 | 2-Piperidinoethyl 4-amino-5-chloro-...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056416(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-acety...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398588(CHEMBL2179582)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at rat 5HT4S receptor expressed in HEK293 cells assessed as increase in cAMP production after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50454556(CHEMBL2115017)
Affinity DataKi:  1.20nMAssay Description:Binding affinity at 5-hydroxytryptamine 4 receptor in rat striatal membranes by [3H]GR-113808 displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM82505(CAS_121881 | NSC_121881 | SB204070)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85135(RS 57639)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85135(RS 57639)
Affinity DataKi:  1.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056411(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-carba...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50056424(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-hydro...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50181844((1R,7aS)-hexahydro-1H-pyrrolizin-1-ylmethyl 4-amin...)
Affinity DataEC50:  1.5nMAssay Description:Agonism at 5HT4 receptor in rat tunica muscularis mucosaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398590(CHEMBL2179583)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]GR113808 from 5HT4 receptor in rat striatal membrane after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Rat)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM50398588(CHEMBL2179582)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at rat 5HT4L receptor expressed in HEK293 cells assessed as increase in cAMP production after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
Displayed 1 to 50 (of 444 total ) | Next | Last >>
Jump to: