Compile Data Set for Download or QSAR
Report error Found 11 of affinity data for UniProtKB/TrEMBL: Q61391
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041062(3-(4-Hydroxy-phenyl)-2-[2-mercaptomethyl-3-(4-meth...)
Affinity DataIC50: 2.5nMAssay Description:In vivo inhibitory potency against Neutral Endopeptidase by measuring the displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50452141(CHEMBL2372595)
Affinity DataIC50: 500nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50027522(2-(2-Carboxy-3-phenyl-propionylamino)-4-methyl-pen...)
Affinity DataIC50: 700nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50027514(2-(2-Carboxymethyl-3-phenyl-propionylamino)-4-meth...)
Affinity DataIC50: 800nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataIC50: 1.00E+3nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50027518((2S)-2-[(2R)-2-[(carboxylatomethyl)amino]-3-phenyl...)
Affinity DataIC50: 2.00E+3nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50027513(2-[2-(2-Carboxy-ethylamino)-3-phenyl-propionylamin...)
Affinity DataIC50: 1.10E+4nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50224343(CHEMBL3350383)
Affinity DataIC50: 1.10E+4nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50027517(CHEMBL2372594)
Affinity DataIC50: 1.80E+4nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50027518((2S)-2-[(2R)-2-[(carboxylatomethyl)amino]-3-phenyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50027516(CHEMBL37879 | 2-(2-Amino-3-phenyl-propionylamino)-...)
Affinity DataIC50: 7.00E+5nMAssay Description:50% Inhibitory potency against enkephalinase from mouse striatum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed