Compile Data Set for Download or QSAR
Report error Found 15 of affinity data for UniProtKB/TrEMBL: Q61214
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50026622(CHEMBL408982)
Affinity DataIC50: 12nMAssay Description:Inhibition of mouse glutathione S-transferase-tagged Dyrk1A expressed in Escherichia coli DH5alpha using NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH peptide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50087427(8-Hydroxy-2-[2-(3-hydroxy-4-methoxy-phenyl)-vinyl]...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of mouse DYRK1A expressed in Escherichia coli after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187069(1-(3,4-dichlorophenyl)-4-(4-hydroxy-3-methoxybenzy...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50145371(2-(2,4-Dihydroxy-benzylcarbamoyl)-8-hydroxy-quinol...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of mouse DYRK1A expressed in Escherichia coli after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187059(1-(3-methoxyphenyl)-3-(5-(pyridin-4-yl)-1,3,4-thia...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187063(N2-(4-bromophenyl)-N4-(furan-2-ylmethyl)quinazolin...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187065(diethyl 4-(4-acetamidophenylamino)quinoline-3,6-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187062(5-(5-(2-(allyloxy)-5-bromobenzylidene)-4-oxo-4,5-d...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187067(2-(5-(2-chlorophenyl)-1H-pyrazol-3-yl)-4-methoxyph...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187060((Z)-3-(2-(4-fluorophenylamino)-4-oxothiazol-5(4H)-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187061(3-ethyl 6-methyl 4-(3-acetylphenylamino)quinoline-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187064(4-(2-methylimidazo[1,2-a]pyrimidin-3-yl)-N-m-tolyl...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187066(4-(4-hydroxy-3-methoxybenzylidene)-1-(3-chlorophen...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Mouse)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50187068(diethyl 4-(3-bromo-4-methylphenylamino)quinoline-3...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed