Compile Data Set for Download or QSAR
Report error Found 12 of affinity data for UniProtKB/TrEMBL: Q53EL6
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50345540(Cryptocaryol A | CHEMBL1784372)
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50345541(Cryptocaryol B | CHEMBL1784373)
Affinity DataEC50:  3.00E+3nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50345542(Cryptocaryol C | CHEMBL1784374)
Affinity DataEC50:  1.60E+3nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50345543(Cryptocaryol D | CHEMBL1784375)
Affinity DataEC50:  1.50E+3nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50345544(Cryptocaryol E | CHEMBL1784376)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50345545(Cryptocaryol F | CHEMBL1784377)
Affinity DataEC50:  3.50E+3nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50345546(Cryptocaryol G | CHEMBL1784378)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50345547(Cryptocaryol H | CHEMBL1784379)
Affinity DataEC50:  1.80E+3nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM36609(Rapamycin C-7, analog 4 | SIROLIMUS | US11603377, ...)
Affinity DataEC50:  50nMAssay Description:Inhibition of TPA-induced degradation of Pdcd4 (amino acid 39-91) expressed in human HEK293 cells assessed as minimum compound concentration required...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50598483(CHEMBL5170759)
Affinity DataEC50:  2.25E+3nMAssay Description:Inhibition of PDCD4 in human HeLa cells tranfected with pCI-neo-luciferase-PDCD4 3'-UTR plasmid assessed as increase in luciferase activity by lucife...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  127nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProgrammed cell death protein 4(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50000298('2-(4-AMINO-PYRROLO[2,3-D]PYRIMIDIN-7-YL)-5-HYDROX...)
Affinity DataIC50: 880nMAssay Description:Stabilization of Pdcd4 expressed in human HEK293 cells assessed as inhibition of TPA-induced degradation by luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed