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TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50611988(CEFTAROLINE | Ceftaroline | T 91825 | T-91825)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity to methicillin sensitive Staphylococcus aureus PBP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50611990(CHEMBL3805841)
Affinity DataIC50: 78nMAssay Description:Inhibition of Staphylococcus aureus PBP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50483327(CEFTOBIPROLE MEDOCARIL)
Affinity DataIC50: 144nMAssay Description:Inhibition of methicillin-susceptible Staphylococcus aureus ATCC 29213 PBP 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50482776(CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...)
Affinity DataIC50: 146nMAssay Description:Binding affinity to methicillin-susceptible Staphylococcus aureus PBP 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50378857(Zeftera | Zevtera | CEFTOBIPROLE)
Affinity DataIC50: 187nMAssay Description:Inhibition of bocillin FL binding to methicillin-susceptible Staphylococcus aureus ATCC 29213 penicillin-binding protein 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50103601(CHEBI:29007 | Ceftriaxone)
Affinity DataIC50: 901nMAssay Description:Inhibition of bocillin FL binding to methicillin-susceptible Staphylococcus aureus ATCC 29213 penicillin-binding protein 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218769(CHEMBL67628)
Affinity DataIC50: 4.94E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218762(CHEMBL306206)
Affinity DataIC50: 5.32E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218764(CHEMBL67669)
Affinity DataIC50: 5.45E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218771(CHEMBL63749)
Affinity DataIC50: 5.52E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218772(CHEMBL66853)
Affinity DataIC50: 5.67E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218763(CHEMBL67946)
Affinity DataIC50: 5.77E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218767(CHEMBL67954)
Affinity DataIC50: 6.50E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218765(CHEMBL66962)
Affinity DataIC50: 6.63E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218773(CHEMBL432719)
Affinity DataIC50: 6.78E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218761(CHEMBL304925)
Affinity DataIC50: 6.78E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218760(CHEMBL304750)
Affinity DataIC50: 7.03E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218768(CHEMBL68222)
Affinity DataIC50: 7.30E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218766(CHEMBL67473)
Affinity DataIC50: 7.80E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed
TargetPutative penicillin-binding protein 2B(Staphylococcus aureus)
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50218770(CHEMBL294507)
Affinity DataIC50: 8.98E+5nMAssay Description:Inhibition of Penicillin-binding protein 1 (PBP1) from Staphylococcus aureusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2018
Entry Details Article
PubMed