Compile Data Set for Download or QSAR
Report error Found 10 of affinity data for UniProtKB/TrEMBL: Q2FXH2
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286770(CHEMBL4171058)
Affinity DataIC50: 640nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286767(CHEMBL4172643)
Affinity DataIC50: 650nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286774(CHEMBL4163140)
Affinity DataIC50: 920nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286768(CHEMBL4171458)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286765(CHEMBL4159778)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286771(CHEMBL4167692)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286775(CHEMBL4174152)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286766(CHEMBL4163450)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286772(CHEMBL4160841)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
TargetLeucine--tRNA ligase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Oxford Drug Design

Curated by ChEMBL
LigandPNGBDBM50286769(CHEMBL4161986)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of Staphylococcus aureus LeuRS expressed in Escherichia coli M15 cells assessed as reduction in ATP consumptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed